SCHEMBL9490891

SCHEMBL9490891

COc1ccc(COc2ccc3c(c2)CCCC3NO)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
TAS1R3 Q7RTX0 1/20 0.47
TAS1R1 Q7RTX1 1/20 0.47
TAS1R2 Q8TE23 1/20 0.47
SPHK2 Q9NRA0 1/20 0.47
SMPD1 P17405 1/20 0.46
MMP1 P03956 1/20 0.46
MMP2 P08253 1/20 0.46
MMP7 P09237 1/20 0.46
MMP9 P14780 1/20 0.46
MMP12 P39900 1/20 0.46
MMP14 P50281 1/20 0.46
MMP15 P51511 1/20 0.46
MMP16 P51512 1/20 0.46
MMP26 Q9NRE1 1/20 0.46
SCN3A Q9NY46 1/20 0.46
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
BDKRB1 P46663 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9488534 0.93 SMPD1 (0.48) SPHK2SMPD1MMP1MMP2MMP7
SCHEMBL9490621 0.88 MAOB (0.52) ALDH1A1TAS1R3TAS1R1TAS1R2SPHK2
SCHEMBL9487573 0.88 TAOK1 (0.53) MMP1MMP2MMP7MMP9MMP12
SCHEMBL9490515 0.86 TAS1R3 (0.56) ALDH1A1TAS1R3TAS1R1TAS1R2MEN1
SCHEMBL9492340 0.84 GAA (0.48) ALDH1A1SCN3ATAOK1MAPT
SCHEMBL9488808 0.80 LIPG (0.57) MMP1MMP2MMP7MMP9MMP12
SCHEMBL22289691 0.80 ADRA1D (0.44) SPHK2ADRA1DADRA1AADRA1BNPC1
SCHEMBL29766272 0.80 ADRA1D (0.44) SPHK2ADRA1DADRA1AADRA1BNPC1
SCHEMBL14378591 0.78 PPARD (0.67)
SCHEMBL9491587 0.78 TAOK1 (0.53) ADRA1DADRA1AADRA1BTAOK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0522000-A1 5-LIPOXYGENASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1993-01-13 EP disclosed
WO-1991014674-A2 5-LIPOXYGENASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1991-10-03 WO disclosed