SCHEMBL9501326

SCHEMBL9501326

N#Cc1cccc2[nH]c(OC(=O)O)cc(=O)c12

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 1/20 0.35
PARP1 P09874 2/20 0.33
GRIA1 P42261 1/20 0.33
CACNG8 Q8WXS5 1/20 0.33
MMP13 P45452 1/20 0.32
CLK1 P49759 2/20 0.32
DYRK1A Q13627 2/20 0.32
CLK2 P49760 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
MCL1 Q07820 1/20 0.31
GPR35 Q9HC97 1/20 0.31
KDM4E B2RXH2 1/20 0.31
GALR3 O60755 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9499661 0.80 IMPDH2 (0.40) PARP1MCL1GPR35KDM4EALDH1A1
SCHEMBL9500387 0.79 FEN1 (0.43) PARP1
SCHEMBL9452237 0.79 HPGD (0.53) GPR35KDM4EALDH1A1GAAHPGD
SCHEMBL9501069 0.77 DAO (0.40)
SCHEMBL9500238 0.76 PARP1 (0.31) PARP1GPR35KDM4EALDH1A1GAA
SCHEMBL9499289 0.76 KDM4E (0.37) PARP1MCL1KDM4EALDH1A1HPGD
SCHEMBL9500319 0.76 CDK1 (0.37) PARP1
SCHEMBL9389922 0.74 DAO (0.46) MAP2K1MCL1
SCHEMBL9499677 0.74 PLA2G2A (0.38) GPR35
SCHEMBL9502885 0.73 PDE2A (0.42) MCL1GPR35KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0303387-B1 KYNURENIC ACID DERIVATIVES USEFUL IN THE TREATMENT OF NEURODEGENERATIVE DISORDERS MERCK SHARP & DOHME LTD. (GB) 1993-04-21 EP claimed