SCHEMBL9502415

SCHEMBL9502415

Cc1ccc(Sc2c(Cl)cc(N3NCC(=O)NC3=O)cc2Cl)cc1C

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.34
GAA P10253 2/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
NOTUM Q6P988 1/20 0.33
MAPK13 O15264 1/20 0.33
MAPK12 P53778 1/20 0.33
MAPK11 Q15759 1/20 0.33
MAPK14 Q16539 1/20 0.33
PKM P14618 1/20 0.33
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
HTR1A P08908 2/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C9 P11712 2/20 0.32
HTR3A P46098 2/20 0.32
MAPT P10636 2/20 0.31
HPGD P15428 2/20 0.31
ALDH1A1 P00352 1/20 0.31
OPRM1 P35372 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9504429 0.88 MEN1 (0.38) KMT2AGAAMEN1LMNANOTUM
SCHEMBL9501160 0.85 LMNA (0.36) KMT2AGAAMEN1LMNAALDH1A1
SCHEMBL9501084 0.85 MEN1 (0.42) KMT2AGAAMEN1LMNANOTUM
SCHEMBL10501494 0.84 KMT2A (0.36) KMT2AGAAMEN1NOTUMPKM
SCHEMBL9500884 0.78 MEN1 (0.37) KMT2AGAAMEN1LMNANOTUM
SCHEMBL10733171 0.74 HTR1A (0.36) KMT2AMEN1CYP1A2CYP3A4HTR1A
SCHEMBL9504425 0.71 NPBWR1 (0.35) LMNAALDH1A1SMN1; SMN2
SCHEMBL7919150 0.70 TSHR (0.38) KMT2AMEN1MAPTALDH1A1
SCHEMBL10502467 0.67 NPC1 (0.40) LMNAMAPTALDH1A1SMN1; SMN2
SCHEMBL2033033 0.67 CYP3A4 (0.47) KMT2AMAPK13MAPK12MAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0154885-B1 SUBSTITUTED 2-PHENYL-HEXAHYDRO-1,2,4-TRIAZINE-2,5-DIONES, METHOD FOR THEIR PREPARATION, THEIR USE AS VETERINARY MEDICINES AND FOR COMBATING PROTOZOES HOECHST AKTIENGESELLSCHAFT (DE) 1989-01-18 EP claimed
US-5188832-A Triazine-dione compounds HOECHST AKTIENGESELLSCHAFT (DE) 1993-02-23 US disclosed