SCHEMBL9508035

SCHEMBL9508035

CN(Cc1ccc(S(=O)(=O)c2ccccc2)cc1)c1cccc2cccc(N)c12

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TYMS P04818 2/20 0.55
HTR6 P50406 5/20 0.42
SCN9A Q15858 1/20 0.39
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
NCOR2 Q9Y618 1/20 0.37
FFAR2 O15552 1/20 0.37
LOX P28300 1/20 0.36
RAB9A P51151 1/20 0.36
CXCR4 P61073 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9965483 0.74 AOC3 (0.52) HDAC3HDAC1HDAC2NCOR2RAB9A
SCHEMBL12083406 0.72 ALDH1A1 (0.59) TYMSHTR6CXCR4L3MBTL1
SCHEMBL4664189 0.71 TYMS (0.46) TYMSHTR6L3MBTL1
SCHEMBL4664193 0.71 TYMS (0.46) TYMSHTR6CXCR4L3MBTL1CRHBP
SCHEMBL9701972 0.71 TYMS (0.53) TYMSHTR6SCN9AFFAR2
SCHEMBL9504568 0.70 TYMS (0.69) TYMSHTR6FFAR2CRHBPCRHR2
SCHEMBL9587756 0.68 TYMS (0.43) TYMSHTR6HDAC3HDAC1HDAC2
SCHEMBL9508662 0.68 TYMS (0.59) TYMSRAB9ACRHBPCRHR2
SCHEMBL1065778 0.67 DHFR (0.59) TYMS
SCHEMBL158288 0.67 HTR6 (0.71) HTR6LOX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0550566-A1 ANTIPROLIFERATIVE SUBSTITUTED NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS (US) 1993-07-14 EP disclosed
WO-1992005153-A1 ANTIPROLIFERATIVE SUBSTITUTED NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1992-04-02 WO disclosed