SCHEMBL9505234

SCHEMBL9505234

CCOC(=O)C1=C(CCl)NC(C)=C(C(=O)OC(C)(C)C)C1c1cccc2c1OCCO2

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.61
MGAM O43451 1/20 0.61
AMY1A P0DUB6 1/20 0.61
SI P14410 1/20 0.61
MGAM2 Q2M2H8 1/20 0.61
CYP2C9 P11712 4/20 0.48
CYP3A4 P08684 3/20 0.48
CYP2C19 P33261 3/20 0.48
LMNA P02545 3/20 0.48
ADORA3 P0DMS8 3/20 0.48
OPRK1 P41145 3/20 0.48
SLC6A2 P23975 3/20 0.48
DRD3 P35462 3/20 0.48
KCNH2 Q12809 3/20 0.48
NR1I2 O75469 2/20 0.48
PGR P06401 2/20 0.48
PDE4D Q08499 2/20 0.48
HTT P42858 1/20 0.48
TBXAS1 P24557 1/20 0.48
KDM4E B2RXH2 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9518606 0.90 GAA (0.64) GAAMGAMAMY1ASIMGAM2
SCHEMBL9502266 0.83 MGAM (0.54) GAAMGAMAMY1ASIMGAM2
SCHEMBL9504261 0.75 MGAM (0.66) GAAMGAMAMY1ASIMGAM2
SCHEMBL7375366 0.73 TBXA2R (0.67) GAACYP2C9CYP3A4CYP2C19LMNA
Oxodipine SCHEMBL332244 0.73 GAA (0.91) GAAMGAMAMY1ASIMGAM2
SCHEMBL9504232 0.72 KDM4E (0.43) GAACYP2C9CYP3A4CYP2C19LMNA
SCHEMBL6589196 0.72 CACNA1F (0.60) CACNA1C
SCHEMBL9513012 0.70 CACNA1C (0.53) GAACYP2C9CYP3A4CYP2C19LMNA
SCHEMBL9504286 0.70 GAA (0.59) GAAMGAMAMY1ASIMGAM2
Hydrochloric Acid SCHEMBL9503007 0.70 MGAM (0.49) GAAMGAMAMY1ASIMGAM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458823-B1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1993-10-13 EP disclosed
US-5245039-A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA (IT) 1993-09-14 US disclosed
WO-1990009376-A1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-23 WO disclosed
EP-0383320-A1 A process for preparation of enantiomerically pure polysubstituted 1,4-dihydropyridines BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-22 EP disclosed