SCHEMBL9506919

SCHEMBL9506919

COc1cc(C)c2c(c1C)CCC2

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 4/20 0.42
HTR2A P28223 1/20 0.37
ALDH1A1 P00352 2/20 0.36
USP2 O75604 1/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
BRD4 O60885 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP3A4 P08684 1/20 0.34
ADRA1A P35348 1/20 0.34
ACHE P22303 2/20 0.33
CASP6 P55212 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
DHFR P00374 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21367505 0.79 ERN1 (0.42) ALOX5ALDH1A1LMNAMAPTL3MBTL1
SCHEMBL18920026 0.77 PNMT (0.41) ALOX5HTR2ALMNA
SCHEMBL31556321 0.75 ALOX5 (0.43) ALOX5HTR2AMEN1KMT2AADRA1A
SCHEMBL8872403 0.75 ERN1 (0.42) ALOX5ALDH1A1LMNAMAPTL3MBTL1
SCHEMBL25647588 0.74 CASP1 (0.43) HTR2AALDH1A1LMNAMEN1KMT2A
SCHEMBL9817570 0.72 ACHE (0.41) ALDH1A1MAPTNPSR1BRD4MEN1
SCHEMBL22596240 0.72 EHMT2 (0.36) ALOX5ALDH1A1MAPTL3MBTL1MEN1
SCHEMBL2722920 0.71 ADRA1A (0.52) ALDH1A1LMNANPSR1MEN1KMT2A
SCHEMBL6314736 0.71 HTR2A (0.36) ALOX5HTR2AALDH1A1LMNAPOLB
SCHEMBL9510782 0.71 ALDH1A1 (0.53) ALOX5ALDH1A1LMNAMAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0295037-B1 PHENOL DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-08-18 EP disclosed
US-5162571-A Phenol derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-11-10 US disclosed
EP-0295037-A2 Phenol derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1988-12-14 EP disclosed