SCHEMBL9508261

SCHEMBL9508261

O=C(CI)Nc1ccc(NOS(=O)(=O)c2cccc3ccccc23)cc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.44
KMT2A Q03164 5/20 0.44
TSHR P16473 1/20 0.41
HTR6 P50406 7/20 0.41
HTR2C P28335 2/20 0.41
HTR2B P41595 2/20 0.41
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
DEGS1 O15121 1/20 0.39
PGR P06401 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9139273 0.80 PGR (0.49) MEN1KMT2ATSHRHTR6ALDH1A1
Ammonia Solution, Strong SCHEMBL28968464 0.79 PGR (0.48) MEN1KMT2ATSHRHTR6ALDH1A1
SCHEMBL8928012 0.78 CA2 (0.48) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL8928011 0.77 TSHR (0.40) TSHRHTR6ALDH1A1
SCHEMBL8919664 0.72 POLB (0.46) MEN1KMT2AALDH1A1
SCHEMBL8960993 0.72 CHAT (0.39) MEN1KMT2ATSHRPGR
SCHEMBL28753722 0.71 KEAP1 (0.49) MEN1KMT2ATSHRHTR6ALDH1A1
SCHEMBL8928013 0.71 MAPT (0.40) MEN1KMT2AHTR6ALDH1A1TP53
SCHEMBL22187492 0.70 CA2 (0.63) PGRRAB9A
SCHEMBL28173820 0.70 F2 (0.52) TSHRHTR6ALDH1A1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0557383-A1 METHOD OF INHIBITING TRANSFORMATION, GROWTH AND METASTASIS OF CELLS IN WHICH PURINE METABOLIC ENZYME ACTIVITY IS ELEVATED AMIRA, INC. (US) 1993-09-01 EP disclosed