SCHEMBL9508330

SCHEMBL9508330

COC(C)(C)c1ccccc1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.41
ACHE P22303 2/20 0.41
GABRA1 P14867 1/20 0.40
GABRB2 P47870 1/20 0.40
TDP1 Q9NUW8 2/20 0.37
CYP3A4 P08684 1/20 0.37
MAPK1 P28482 1/20 0.36
CASR P41180 1/20 0.35
ALDH1A1 P00352 4/20 0.34
CA2 P00918 3/20 0.33
CA1 P00915 2/20 0.33
CA7 P43166 2/20 0.33
CA9 Q16790 2/20 0.33
HSP90AA1 P07900 1/20 0.33
ALOX15 P16050 1/20 0.33
ESR1 P03372 1/20 0.33
GAA P10253 1/20 0.32
CYP2A6 P11509 2/20 0.31
TRPA1 O75762 1/20 0.31
ATM Q13315 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29947075 0.85 MAPK1 (0.42) TSHRGABRA1GABRB2TDP1MAPK1
SCHEMBL6900861 0.85 MAPK1 (0.42) TSHRGABRA1GABRB2TDP1MAPK1
SCHEMBL10593629 0.83 TSHR (0.43) TSHRACHEGABRA1GABRB2TDP1
SCHEMBL2270593 0.82 TRPA1 (0.43) TSHRACHEGABRA1GABRB2TDP1
SCHEMBL9504882 0.81 GABRA1 (0.45) TSHRACHEGABRA1GABRB2TDP1
SCHEMBL11106181 0.81 TSHR (0.41) TSHRACHEGABRA1GABRB2TDP1
SCHEMBL8740212 0.79 ALDH1A1 (0.52) TSHRACHEGABRA1GABRB2TDP1
SCHEMBL13408217 0.79 TSHR (0.39) TSHRACHEGABRA1GABRB2TDP1
SCHEMBL17507508 0.79 ACHE (0.39) TSHRACHEGABRA1GABRB2TDP1
SCHEMBL1318701 0.79 TSHR (0.39) TSHRACHEGABRA1GABRB2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9566290-B2 Boron-containing small molecules ANACOR PHARMACEUTICALS, INC. (US) 2017-02-14 US disclosed
EP-2982672-A1 Hypervalent iodine CF2CF2X reagents and their use ETH Zurich (CH) 2016-02-10 EP disclosed
EP-2021330-B1 BENZIMIDAZOLE MODULATORS OF VR1 JANSSEN PHARMACEUTICA NV (BE) 2010-09-22 EP disclosed
US-7388021-B2 Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions BRISTOL MYERS SQUIBB COMPANY (US) 2008-06-17 US disclosed
EP-0261962-B1 PROCESS FOR PRODUCING PROPYLENE BLOCK COPOLYMER MITSUBISHI PETROCHEMICAL CO., LTD. (JP) 1993-07-28 EP disclosed
EP-0261962-A2 Process for producing propylene block copolymer MITSUBISHI PETROCHEMICAL CO., LTD. (JP) 1988-03-30 EP disclosed