SCHEMBL9513601

SCHEMBL9513601

COc1ccc2[nH]cc(OCCN)c2c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.61
HTR1A P08908 5/20 0.61
HTR2C P28335 4/20 0.61
HTR1B P28222 4/20 0.61
HTR1D P28221 3/20 0.61
CYP1A2 P05177 2/20 0.61
MAPT P10636 1/20 0.61
TSHR P16473 1/20 0.61
NFKB1 P19838 1/20 0.61
HTR7 P34969 1/20 0.61
HTR6 P50406 1/20 0.61
HTR4 Q13639 1/20 0.61
TRPM8 Q7Z2W7 1/20 0.61
HTR2B P41595 4/20 0.60
BLM P54132 1/20 0.59
PMP22 Q01453 1/20 0.59
NPSR1 Q6W5P4 1/20 0.59
GPR84 Q9NQS5 2/20 0.55
CYP2D6 P10635 1/20 0.50
MEN1 O00255 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3563693 0.83 HTR6 (0.63) HTR2AHTR1AHTR2CHTR1BHTR1D
SCHEMBL28337310 0.81 GPR84 (0.64) HTR2AHTR1AHTR2CHTR1BHTR1D
SCHEMBL4489769 0.76 NR4A2 (0.57) HTR1ACYP1A2MAPTHTR2BBLM
5-Methoxytryptamine SCHEMBL41982 0.76 HTR1A (1.00) HTR2AHTR1AHTR2CHTR1BHTR1D
5-Methoxytryptamine SCHEMBL29390103 0.76 HTR1A (1.00) HTR2AHTR1AHTR2CHTR1BHTR1D
SCHEMBL3976318 0.75 HTR2B (1.00) HTR2AHTR1AHTR2CHTR1BHTR1D
5-Methoxytryptamine SCHEMBL130877 0.75 HTR1A (0.97) HTR2AHTR1AHTR2CHTR1BHTR1D
5-Methoxytryptamine SCHEMBL1322980 0.75 NPSR1 (1.00) HTR2AHTR1AHTR2CHTR1BHTR1D
5-Methoxytryptamine SCHEMBL31109114 0.75 NPSR1 (1.00) HTR2AHTR1AHTR2CHTR1BHTR1D
5-Methoxytryptamine SCHEMBL26617456 0.75 HTR1A (0.97) HTR2AHTR1AHTR2CHTR1BHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5227488-A AZA SPIRO DECANE AND USE THEREOF IN TREATING CNS DISORDERS NOVO NORDISK A/S (DK) 1993-07-13 US disclosed
EP-0495826-A1 INDOLE DERIVATIVES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1992-07-29 EP disclosed
WO-1991004973-A1 INDOLE DERIVATIVES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1991-04-18 WO disclosed