SCHEMBL9516072

SCHEMBL9516072

CC(C)c1cc(C2CCCCC2)cc(-c2ccc(F)cc2)c1O

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.44
HMGCR P04035 5/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C9 P11712 1/20 0.39
GCGR P47871 2/20 0.38
MAPK14 Q16539 1/20 0.38
DHODH Q02127 1/20 0.35
HSP90AA1 P07900 2/20 0.35
HSP90AB1 P08238 2/20 0.35
PTGDR Q13258 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
PTGS2 P35354 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27698484 0.80 CA1 (0.48) CYP3A4CA1CA2
SCHEMBL9512239 0.75 CA1 (0.53) HMGCRCYP3A4GCGRHSP90AA1HSP90AB1
SCHEMBL8780176 0.74 GABRA1 (0.50) HMGCRGCGRHSP90AA1HSP90AB1CA1
SCHEMBL27579607 0.73 GABRA1 (0.43) CYP2C9HSP90AA1HSP90AB1CA1CA2
SCHEMBL9199239 0.73 CA1 (0.41) HMGCRCYP3A4GCGRHSP90AA1HSP90AB1
SCHEMBL9622089 0.73 GABRA1 (0.43) CYP2C9HSP90AA1HSP90AB1CA1CA2
SCHEMBL27579601 0.73 GABRA1 (0.43) CYP2C9HSP90AA1HSP90AB1PTGDRPTGDR2
SCHEMBL8780227 0.72 HMGCR (0.50) HMGCRCYP2C9GCGRMAPK14DHODH
SCHEMBL9514348 0.71 CA1 (0.47) HMGCRHSP90AA1CA1CA2PTGS2
SCHEMBL9516053 0.71 CA1 (0.39) CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0341681-B1 6-Phenoxymethyl-4-hydroxytetrahydropyran-2-ones and 6-thiophenoxymethyl-4-hydroxytetrahydropyran-2-ones, the corresponding dihydrocarboxylic-acid derivatives, salts and esters, process for preparing these compounds, their use as medicines, pharmaceutical compositions and phenols and thiophenols HOECHST AG (DE) 1993-12-29 EP disclosed
US-5166171-A Compounds for treatment of artheriosclerosis and hypercholesterolemia HOECHST AKTIENGESELLSCHAFT (DE) 1992-11-24 US disclosed
EP-0341681-A2 6-Phenoxymethyl-4-hydroxytetrahydropyran-2-ones and 6-thiophenoxymethyl-4-hydroxytetrahydropyran-2-ones, the corresponding dihydrocarboxylic-acid derivatives, salts and esters, process for preparing these compounds, their use as medicines, pharmaceutical compositions and phenols and thiophenols HOECHST AKTIENGESELLSCHAFT (DE) 1989-11-15 EP disclosed