SCHEMBL9517088

SCHEMBL9517088

O=CC(c1ccc(F)cc1)S(=O)(=O)NC(=O)c1ccc(COC(=O)c2ccccc2)nc1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 5/20 0.38
CXCR1 P25024 3/20 0.38
EPHX2 P34913 5/20 0.38
CASP3 P42574 4/20 0.38
KMT2A Q03164 1/20 0.38
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
CYP2J2 P51589 1/20 0.37
BCL2L1 Q07817 1/20 0.36
MCL1 Q07820 1/20 0.36
P4HTM Q9NXG6 2/20 0.35
MAPT P10636 1/20 0.35
PTGS2 P35354 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9515607 0.88 EPHX2 (0.40) CXCR2CXCR1EPHX2CASP3CYP2C9
SCHEMBL9517908 0.85 CXCR1 (0.39) CXCR2CXCR1EPHX2CASP3CYP2C9
SCHEMBL9518019 0.83 MEN1 (0.39) CXCR2CXCR1EPHX2CASP3KMT2A
SCHEMBL9517093 0.82 P4HTM (0.39) CXCR2CXCR1EPHX2KMT2ACYP2C9
SCHEMBL9517229 0.80 POLB (0.38) CXCR2CXCR1CASP3P4HTMMAPT
SCHEMBL9519643 0.79 GRM5 (0.39) CXCR2CXCR1CASP3P4HTM
SCHEMBL9517259 0.78 EGFR (0.39) EPHX2CASP3P4HTM
SCHEMBL9517222 0.78 TRPM8 (0.38) EPHX2CASP3P4HTM
SCHEMBL9515729 0.78 BCL2L1 (0.40) CXCR2CASP3KMT2ABCL2L1MCL1
SCHEMBL9516087 0.78 BCL2L1 (0.38) CXCR2EPHX2CASP3BCL2L1MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0567997-A1 4- or 5-(sulf)imido- and (sulfon)amidopyridines and their pyridine-N-oxides, process for their preparation and their use as pharmaceutical HOECHST AKTIENGESELLSCHAFT (DE) 1993-11-03 EP disclosed