SCHEMBL9521157

SCHEMBL9521157

N#Cc1ccc(C(=O)N2CC3CC(CN(Cc4ccccc4)C3)C2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
FAAH O00519 1/20 0.49
PRKAB2 O43741 1/20 0.48
PRKAG1 P54619 1/20 0.48
PRKAA2 P54646 1/20 0.48
PRKAA1 Q13131 1/20 0.48
PRKAG3 Q9UGI9 1/20 0.48
PRKAG2 Q9UGJ0 1/20 0.48
PRKAB1 Q9Y478 1/20 0.48
CHRNB2 P17787 1/20 0.47
CHRNB4 P30926 1/20 0.47
CHRNA3 P32297 1/20 0.47
CHRNA7 P36544 1/20 0.47
CHRNA4 P43681 1/20 0.47
CHRM4 P08173 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2D6 P10635 1/20 0.47
KDM4E B2RXH2 1/20 0.46
USP2 O75604 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9521948 0.84 ALDH1A1 (0.50) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL9521802 0.84 SIGMAR1 (0.50) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
Ambasilide SCHEMBL427931 0.84 HSD11B1 (0.53) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL9521359 0.84 KMT2A (0.58) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA7
Ambasilide SCHEMBL246531 0.84 HSD11B1 (0.53) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL13149337 0.81 ALDH1A1 (0.70) ALDH1A1FAAHSMN1; SMN2KDM4ETSHR
SCHEMBL9520996 0.81 CYP2D6 (0.61) ALDH1A1FAAHCHRNB2CHRNB4CHRNA3
SCHEMBL9523517 0.81 ALDH1A1 (0.51) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL10409272 0.81 SIGMAR1 (0.68) FAAHPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL9520394 0.80 HTT (0.50) ALDH1A1PRKAB2PRKAG1PRKAA2PRKAA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308843-B1 Bispidin derivatives as class III antiarrhythmics BASF AG (DE) 1993-12-15 EP disclosed
US-4959373-A Bispidine derivatives as class III antiarrhythmic agents BASF AKTIENGESELLSCHAFT (DE) 1990-09-25 US disclosed
EP-0308843-A2 Bispidin derivatives as class III antiarrhythmics BASF Aktiengesellschaft (DE) 1989-03-29 EP disclosed