SCHEMBL9520394

SCHEMBL9520394

CC(=O)Nc1ccc(C(=O)N2CC3CC(CN(Cc4ccccc4)C3)C2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.50
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 1/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
PRKAB2 O43741 1/20 0.47
PRKAG1 P54619 1/20 0.47
PRKAA2 P54646 1/20 0.47
PRKAA1 Q13131 1/20 0.47
PRKAG3 Q9UGI9 1/20 0.47
PRKAG2 Q9UGJ0 1/20 0.47
PRKAB1 Q9Y478 1/20 0.47
GRIN2B Q13224 1/20 0.47
CYP2C19 P33261 1/20 0.46
CHRNB2 P17787 1/20 0.46
CHRNB4 P30926 1/20 0.46
CHRNA3 P32297 1/20 0.46
CHRNA7 P36544 1/20 0.46
CHRNA4 P43681 1/20 0.46
TSHR P16473 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10410772 0.90 POLB (0.54) ALDH1A1KDM4EMEN1KMT2ACYP2C19
SCHEMBL9521948 0.85 ALDH1A1 (0.50) ALDH1A1KDM4EMEN1KMT2ACHRNB2
SCHEMBL9523570 0.85 PKM (0.50) HTTALDH1A1MEN1KMT2APRKAB2
Ambasilide SCHEMBL246531 0.83 HSD11B1 (0.53) ALDH1A1KDM4EMEN1KMT2ACHRNB2
SCHEMBL9521359 0.83 KMT2A (0.58) HTTALDH1A1KDM4EMEN1KMT2A
Ambasilide SCHEMBL427931 0.83 HSD11B1 (0.53) ALDH1A1KDM4EMEN1KMT2ACHRNB2
SCHEMBL9521802 0.83 SIGMAR1 (0.50) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL9523517 0.82 ALDH1A1 (0.51) ALDH1A1KDM4EMEN1KMT2ACHRNB2
SCHEMBL9520996 0.82 CYP2D6 (0.61) HTTALDH1A1KDM4EMEN1KMT2A
SCHEMBL9521157 0.80 ALDH1A1 (0.54) ALDH1A1KDM4EPRKAB2PRKAG1PRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-1102078-A None JP disclosed
EP-0308843-B1 Bispidin derivatives as class III antiarrhythmics BASF AG (DE) 1993-12-15 EP disclosed
US-4959373-A Bispidine derivatives as class III antiarrhythmic agents BASF AKTIENGESELLSCHAFT (DE) 1990-09-25 US disclosed
JP-H01102078-A BISPIDINE DERIVATIVE AND ANTIARRHYTHMIC AGENT CONTAINING THE SAME BASF AG 1989-04-19 JP disclosed
EP-0308843-A2 Bispidin derivatives as class III antiarrhythmics BASF Aktiengesellschaft (DE) 1989-03-29 EP disclosed