SCHEMBL9522078

SCHEMBL9522078

O=C(O)C/C=C/C=C(c1ccc(Cl)cc1)c1ccc(Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
CES2 O00748 2/20 0.41
CES1 P23141 2/20 0.41
GSK3B P49841 2/20 0.40
SRD5A2 P31213 1/20 0.40
ERCC5 P28715 1/20 0.40
FEN1 P39748 1/20 0.40
MAPT P10636 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
PAM P19021 1/20 0.38
PTAFR P25105 1/20 0.38
TBXA2R P21731 1/20 0.37
TBXAS1 P24557 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9519681 1.00 ALOX15 (0.44) ALOX15TSHRCES2CES1GSK3B
SCHEMBL9521627 0.84 PAM (0.50) ALOX15TSHRCES2CES1GSK3B
SCHEMBL9520140 0.84 PAM (0.50) ALOX15TSHRCES2CES1GSK3B
SCHEMBL9521054 0.83 CES2 (0.41) ALOX15CES2CES1MAPTALDH1A1
SCHEMBL9519790 0.83 KMT2A (0.44) CES2CES1GSK3BSRD5A2MAPT
SCHEMBL9521278 0.81 SMN1; SMN2 (0.46) TSHRGSK3BERCC5FEN1MAPT
SCHEMBL9519281 0.81 ERCC5 (0.45) ERCC5FEN1MAPTALDH1A1PAM
SCHEMBL9520834 0.81 ERCC5 (0.45) ERCC5FEN1MAPTALDH1A1PAM
SCHEMBL9521346 0.79 CA1 (0.49) CES2CES1GSK3BMAPTALDH1A1
SCHEMBL9421096 0.78 BCL2L1 (0.41) ALOX15TSHRCES2CES1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0299379-B1 PENTADIENAMIDE PAF-ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
EP-0299379-A1 Pentadienamide PAF-antagonists F. HOFFMANN-LA ROCHE AG (CH) 1989-01-18 EP disclosed