SCHEMBL9522136

SCHEMBL9522136

COc1ccc(/C(=C/C=O)c2ccccc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.59
CES1 P23141 2/20 0.59
MAPT P10636 3/20 0.50
ALDH1A1 P00352 3/20 0.50
KDM4E B2RXH2 3/20 0.50
HPGD P15428 2/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
MEN1 O00255 1/20 0.49
HSPD1 P10809 1/20 0.49
TNFRSF1A P19438 1/20 0.49
MAOB P27338 1/20 0.49
HSPE1 P61604 1/20 0.49
KMT2A Q03164 1/20 0.49
CYP1B1 Q16678 1/20 0.49
BCHE P06276 1/20 0.49
CYP3A4 P08684 1/20 0.49
NFKB1 P19838 1/20 0.49
NFKB2 Q00653 1/20 0.49
RELA Q04206 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9522133 1.00 CES2 (0.59) CES2CES1MAPTALDH1A1KDM4E
SCHEMBL9522139 1.00 CES2 (0.59) CES2CES1MAPTALDH1A1KDM4E
SCHEMBL8564034 0.93 ALDH1A1 (0.57) CES2CES1MAPTALDH1A1KDM4E
SCHEMBL7056287 0.89 CES2 (0.62) CES2CES1MAPTALDH1A1KDM4E
SCHEMBL9520429 0.85 MTNR1A (0.57) CES2CES1ALDH1A1MEN1MAOB
SCHEMBL9520437 0.85 MTNR1A (0.57) CES2CES1ALDH1A1MEN1MAOB
SCHEMBL9520444 0.85 MTNR1A (0.57) CES2CES1ALDH1A1MEN1MAOB
SCHEMBL24495087 0.84 NFE2L2 (0.50) CES2CES1MAPTALDH1A1KDM4E
SCHEMBL9522620 0.83 TBXAS1 (0.58) ALDH1A1KDM4EKMT2ACYP1B1NPC1
SCHEMBL9519338 0.83 TBXAS1 (0.58) ALDH1A1KDM4EKMT2ACYP1B1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0299379-B1 PENTADIENAMIDE PAF-ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
US-4975438-A ANTICOAGULANT HOFFMANN-LA ROCHE INC. (US) 1990-12-04 US disclosed
EP-0299379-A1 Pentadienamide PAF-antagonists F. HOFFMANN-LA ROCHE AG (CH) 1989-01-18 EP disclosed
US-4788206-A CARDIOVASCULAR DISORDERS, PLATELETS HOFFMANN-LA ROCHE INC. (US) 1988-11-29 US disclosed