SCHEMBL9523570

SCHEMBL9523570

CS(=O)(=O)Nc1ccc(C(=O)N2CC3CC(CN(Cc4ccccc4)C3)C2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
LMNA P02545 2/20 0.50
ALDH1A1 P00352 1/20 0.50
GAA P10253 1/20 0.50
MAPK1 P28482 1/20 0.50
GRIN2B Q13224 1/20 0.48
ADRB2 P07550 1/20 0.48
ADRB1 P08588 1/20 0.48
ADRB3 P13945 1/20 0.48
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA7 P43166 1/20 0.45
CA9 Q16790 1/20 0.45
CA14 Q9ULX7 1/20 0.45
HPGD P15428 1/20 0.43
HTT P42858 1/20 0.43
CHRNB2 P17787 1/20 0.43
CHRNB4 P30926 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9520394 0.85 HTT (0.50) ALDH1A1GRIN2BHTTCHRNB2CHRNB4
Ambasilide SCHEMBL6385706 0.83 ALDH1A1 (0.47) SMN1; SMN2LMNAALDH1A1MAPK1MEN1
SCHEMBL9521948 0.83 ALDH1A1 (0.50) SMN1; SMN2LMNAALDH1A1MAPK1CHRNB2
SCHEMBL7034748 0.82 HTT (0.53) SMN1; SMN2LMNAALDH1A1MAPK1HPGD
Hydrochloric Acid SCHEMBL8781292 0.82 LMNA (0.70) PKMSMN1; SMN2LMNAALDH1A1GAA
SCHEMBL9521802 0.80 SIGMAR1 (0.50) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
Ambasilide SCHEMBL246531 0.80 HSD11B1 (0.53) SMN1; SMN2LMNAALDH1A1MAPK1CA12
SCHEMBL9521359 0.80 KMT2A (0.58) SMN1; SMN2LMNAALDH1A1MAPK1HPGD
Ambasilide SCHEMBL427931 0.80 HSD11B1 (0.53) SMN1; SMN2LMNAALDH1A1MAPK1CA12
SCHEMBL9520996 0.80 CYP2D6 (0.61) PKMSMN1; SMN2LMNAALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308843-B1 Bispidin derivatives as class III antiarrhythmics BASF AG (DE) 1993-12-15 EP disclosed