SCHEMBL9524288

SCHEMBL9524288

Cc1ccccc1C(=CCCBr)c1ccncc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.46
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
MAPK1 P28482 1/20 0.40
TYK2 P29597 1/20 0.40
SLC6A1 P30531 3/20 0.40
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
CYP19A1 P11511 1/20 0.36
CYP11B2 P19099 1/20 0.36
ALDH1A1 P00352 3/20 0.35
TBXAS1 P24557 3/20 0.35
MAPT P10636 1/20 0.34
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9524284 1.00 L3MBTL1 (0.46) L3MBTL1NPC1RAB9AMAPK1TYK2
SCHEMBL9528603 0.81 CYP19A1 (0.50) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9528596 0.81 CYP19A1 (0.50) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL30331009 0.75 CYP19A1 (0.61) L3MBTL1NPC1RAB9AMAPK1TYK2
SCHEMBL7917518 0.74 SLC6A1 (0.44) L3MBTL1NPC1RAB9ASLC6A1CYP1A2
SCHEMBL7928727 0.74 SLC6A1 (0.44) L3MBTL1NPC1RAB9ASLC6A1CYP1A2
SCHEMBL10285292 0.73 L3MBTL1 (0.55) L3MBTL1NPC1RAB9AMAPK1TYK2
SCHEMBL9524272 0.72 TBXAS1 (0.40) SLC6A1TBXAS1
SCHEMBL9524274 0.72 TBXAS1 (0.40) SLC6A1TBXAS1
SCHEMBL10406652 0.71 RAB9A (0.38) NPC1RAB9ASLC6A1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0231996-B1 NOVEL AMINO ACID DERIVATIVES NOVO NORDISK A/S (DK) 1993-10-06 EP disclosed
US-4931450-A Amino acid derivatives NOVO INDUSTRI A/S (DK) 1990-06-05 US disclosed
EP-0231996-A2 Novel amino acid derivatives NOVO NORDISK A/S (DK) 1987-08-12 EP disclosed