SCHEMBL9525948

SCHEMBL9525948

O=C(CCNS(=O)(=O)c1cccc2ccccc12)ONCCN(C(=O)c1cncc(Br)c1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKD3 O94806 3/20 0.40
PRKCG P05129 3/20 0.40
PRKCB P05771 3/20 0.40
PRKCA P17252 3/20 0.40
PRKCH P24723 3/20 0.40
PRKCI P41743 3/20 0.40
PRKCE Q02156 3/20 0.40
PRKCQ Q04759 3/20 0.40
PRKCZ Q05513 3/20 0.40
PRKCD Q05655 3/20 0.40
PRKD1 Q15139 3/20 0.40
PRKACA P17612 2/20 0.40
PRKACG P22612 2/20 0.40
PRKACB P22694 2/20 0.40
P2RX7 Q99572 1/20 0.37
NPY5R Q15761 2/20 0.37
EGFR P00533 1/20 0.37
MAPK1 P28482 1/20 0.36
CYP3A4 P08684 3/20 0.35
SCN1A P35498 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9524780 0.84 FLT3 (0.43) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL9525433 0.73 EPHX1 (0.45) NPY5RSMN1; SMN2KDM4EALDH1A1CYP1A2
SCHEMBL9525706 0.73 CYP1A2 (0.41) SMN1; SMN2ALDH1A1CYP1A2CYP2C19MEN1
SCHEMBL9525362 0.73 BLM (0.43) MAPK1CYP3A4SMN1; SMN2ALDH1A1CYP1A2
SCHEMBL9524919 0.72 HTT (0.51) EGFRMAPK1SMN1; SMN2KDM4EALDH1A1
SCHEMBL9525284 0.72 ALDH1A1 (0.40) EGFRMAPK1SMN1; SMN2KDM4EALDH1A1
SCHEMBL9525530 0.72 HTT (0.46) EGFRMAPK1CYP3A4SMN1; SMN2ALDH1A1
SCHEMBL9524016 0.71 ALDH1A1 (0.41) SMN1; SMN2KDM4EALDH1A1CYP1A2CYP2C19
Hydrochloric Acid SCHEMBL9528526 0.71 SLC6A9 (0.38) P2RX7NPY5RCYP3A4SCN1ASCN2A
SCHEMBL9525975 0.71 SMN1; SMN2 (0.43) MAPK1SMN1; SMN2ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed