SCHEMBL9525213

SCHEMBL9525213

CSc1nc(-c2ccccc2)c(-c2ccccc2)n1COC(C)[Si](C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 2/20 0.44
MAPK14 Q16539 13/20 0.41
MAPK13 O15264 4/20 0.40
MAPK12 P53778 4/20 0.40
MAPK11 Q15759 4/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
LMNA P02545 1/20 0.36
FAAH O00519 1/20 0.35
PTGS1 P23219 2/20 0.34
PTGS2 P35354 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9525207 0.78 MAPK14 (0.43) ALDH1A1KDM4EMAPK14MAPK13MAPK12
SCHEMBL9370457 0.75 FAAH (0.41) ALDH1A1KDM4EL3MBTL1FAAH
SCHEMBL9370600 0.71 PTGS2 (0.50) ALDH1A1MAPK14MAPK13MAPK12MAPK11
SCHEMBL9369651 0.71 FAAH (0.40) FAAH
SCHEMBL9539522 0.70 NPSR1 (0.50) ALDH1A1KDM4EL3MBTL1LMNA
SCHEMBL4838002 0.68 ALDH1A1 (0.32) ALDH1A1KDM4EFAAH
SCHEMBL7925236 0.64 PPARG (0.39) ALDH1A1KDM4EL3MBTL1LMNA
SCHEMBL13937116 0.62 LMNA (0.60) ALDH1A1KDM4EL3MBTL1LMNA
SCHEMBL13587979 0.62 MEN1 (0.47) ALDH1A1KDM4EMAPK14FAAH
SCHEMBL10967698 0.62 ALDH1A1 (0.49) ALDH1A1KDM4EL3MBTL1LMNAPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993001184-A1 IMIDAZOLES INHIBITORS AS ACAT AND THROMBOXANE TXA2 RHONE-POULENC RORER LIMITED (GB) 1993-01-21 WO disclosed
EP-0522887-A1 Imidazoles as ACAT- and thromboxane TxA2 inhibitors RHONE-POULENC RORER LIMITED (GB) 1993-01-13 EP disclosed