SCHEMBL9525834

SCHEMBL9525834

CCOc1cc(OCC)c(Br)c(-c2ccc(C#N)c(=O)[nH]2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.44
ALDH1A1 P00352 4/20 0.44
GLA P06280 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
GAA P10253 1/20 0.44
IDH1 O75874 2/20 0.37
PDE5A O76074 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
MDM2 Q00987 1/20 0.35
AR P10275 2/20 0.35
MAPT P10636 2/20 0.35
HSD17B10 Q99714 2/20 0.35
ESR2 Q92731 1/20 0.35
PDE3B Q13370 2/20 0.34
PDE3A Q14432 2/20 0.34
PIM1 P11309 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9702558 0.80 ALDH1A1 (0.41) KDM4EALDH1A1GLAL3MBTL1GAA
SCHEMBL7371784 0.79 KDM4E (0.60) KDM4EALDH1A1GLAL3MBTL1GAA
SCHEMBL7646365 0.78 PDE5A (0.50) KDM4EALDH1A1GLAL3MBTL1GAA
SCHEMBL9529353 0.75 CYP2C9 (0.34) KDM4EALDH1A1PDE5AMAPTHSD17B10
SCHEMBL9526090 0.73 KDM4E (0.74) KDM4EALDH1A1GLAL3MBTL1GAA
SCHEMBL9526882 0.73 ALDH1A1 (0.44) KDM4EALDH1A1GLAL3MBTL1GAA
SCHEMBL9702581 0.73 ALDH1A1 (0.44) KDM4EALDH1A1GLAL3MBTL1GAA
SCHEMBL9701860 0.72 KDM4E (0.55) KDM4EALDH1A1GLAL3MBTL1GAA
SCHEMBL9701620 0.71 KDM4E (0.57) KDM4EALDH1A1GLAL3MBTL1GAA
SCHEMBL7647544 0.71 ALDH1A1 (0.54) KDM4EALDH1A1GLAL3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0550576-A1 PHENYLPYRIDINOL DERIVATIVES AS MEDICAMENTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1993-07-14 EP disclosed
WO-1992006085-A1 PHENYLPYRIDINOL DERIVATIVES AS MEDICAMENTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1992-04-16 WO disclosed