SCHEMBL9528273

SCHEMBL9528273

COc1cc(OCCOC(=O)NCCNc2ccccc2)cc(OC)c1OC

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.52
BRD4 O60885 1/20 0.52
LMNA P02545 1/20 0.50
TP53 P04637 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
NPC1 O15118 3/20 0.46
RAB9A P51151 2/20 0.46
TSHR P16473 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ALDH1A1 P00352 2/20 0.45
GAA P10253 1/20 0.45
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
MEN1 O00255 3/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CASR P41180 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9528098 0.83 NPC1 (0.66) KMT2ALMNATP53NPC1RAB9A
SCHEMBL9527973 0.78 NPC1 (0.56) KMT2ALMNATP53NPSR1NPC1
SCHEMBL10182137 0.72 MTNR1A (0.50) KMT2ALMNANPC1RAB9AALDH1A1
SCHEMBL9407487 0.72 CTSK (0.46) KMT2ALMNANPSR1NPC1RAB9A
SCHEMBL9407494 0.72 GAA (0.58) KMT2ALMNANPC1RAB9ASMN1; SMN2
SCHEMBL17550873 0.71 RAB9A (0.59) KMT2ALMNATP53NPC1RAB9A
SCHEMBL7998297 0.69 RAB9A (0.60) KMT2ALMNATP53NPC1RAB9A
SCHEMBL17864863 0.68 NPC1 (0.68) KMT2ALMNATP53NPSR1NPC1
SCHEMBL17550880 0.68 SMN1; SMN2 (0.55) KMT2ALMNATP53NPC1RAB9A
SCHEMBL19750482 0.68 RAB9A (0.55) KMT2ALMNATP53NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed