SCHEMBL9530049

SCHEMBL9530049

COc1ccc2c(CCN3CCN(C(=O)c4ccccc4)C(CC(=O)O)C3=O)c[nH]c2c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.45
MAPT P10636 1/20 0.45
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
ACHE P22303 2/20 0.42
HTR6 P50406 1/20 0.42
HTR2A P28223 1/20 0.41
CDK4 P11802 1/20 0.41
CCND1 P24385 1/20 0.41
HTR1A P08908 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
HPGD P15428 2/20 0.41
DRD4 P21917 1/20 0.41
TSHR P16473 1/20 0.40
RECQL P46063 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9529850 0.93 NPC1 (0.49) KMT2AMEN1MAPTACHEHTR2A
SCHEMBL10491367 0.91 KMT2A (0.42) KMT2AMEN1MAPTMTNR1AMTNR1B
Acetic Acid SCHEMBL10491372 0.91 MTNR1A (0.45) KMT2AMEN1MAPTMTNR1AMTNR1B
SCHEMBL9529587 0.89 PDE4D (0.40) KMT2AACHEHTR2ACDK4CCND1
SCHEMBL10491427 0.85 SLC6A4 (0.46) KMT2AMEN1MAPTACHEHTR2A
Acetic Acid SCHEMBL10491431 0.84 RAB9A (0.48) KMT2AMEN1MAPTMTNR1AMTNR1B
SCHEMBL9529052 0.82 LMNA (0.44) KMT2AMEN1MAPTHTR6HPGD
SCHEMBL10491405 0.82 KMT2A (0.46) KMT2AACHEHPGDSMN1; SMN2
Acetic Acid SCHEMBL10491411 0.80 HPGD (0.40) MAPTACHEHTR2ACDK4CCND1
SCHEMBL10491383 0.80 SMN1; SMN2 (0.48) KMT2AMEN1MAPTHTR2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0287468-B1 17-AZA-20,21-DINOREBURNAMENINE DERIVATIVES, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION, THEIR USE AS MEDICAMENTS AND COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1993-03-10 EP disclosed
EP-0287468-A2 17-Aza-20,21-dinoreburnamenine derivatives, process and intermediates for their preparation, their use as medicaments and compositions containing them ROUSSEL-UCLAF (FR) 1988-10-19 EP disclosed