SCHEMBL9532147

SCHEMBL9532147

COc1ccccc1CCc1ccccc1C(=NO)c1cccnc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.44
CYP3A4 P08684 4/20 0.44
CYP2D6 P10635 4/20 0.44
CYP1A1 P04798 1/20 0.44
CYP1B1 Q16678 1/20 0.44
KMT2A Q03164 3/20 0.43
MAPT P10636 2/20 0.43
CAPN1 P07384 1/20 0.43
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
MEN1 O00255 2/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HTR1A P08908 2/20 0.41
DRD2 P14416 2/20 0.41
USP2 O75604 3/20 0.40
ALOX15 P16050 3/20 0.40
CYP2C19 P33261 3/20 0.40
HSD17B10 Q99714 3/20 0.40
CLK4 Q9HAZ1 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9528143 0.92 CYP1A2 (0.42) CYP1A2CYP3A4CYP2D6CYP1A1CYP1B1
SCHEMBL9529772 0.89 SGMS2 (0.47) KMT2AMAPTSMN1; SMN2HTR1ADRD2
SCHEMBL9527826 0.87 MAPK1 (0.53) CYP1A2CYP3A4CYP2D6CYP1A1CYP1B1
SCHEMBL10407862 0.86 HTR1A (0.46) CYP1A2CYP3A4CYP2D6CYP1A1CYP1B1
SCHEMBL9532132 0.85 KMT2A (0.51) KMT2AHTR1ADRD2USP2ALDH1A1
SCHEMBL9529147 0.84 NOTUM (0.44) KMT2AMAPTMEN1LMNASMN1; SMN2
SCHEMBL9528361 0.82 ALDH1A1 (0.50) CYP1A2CYP2D6KMT2AMAPTMEN1
SCHEMBL9528579 0.82 ALDH1A1 (0.53) KMT2AMAPTMEN1LMNASMN1; SMN2
SCHEMBL10407323 0.82 ABCB1 (0.61) CYP1A2CYP3A4CYP2D6CYP1A1CYP1B1
SCHEMBL9529759 0.81 KMT2A (0.43) CYP1A2KMT2AMAPTLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0366006-B1 PYRIDYLKETOXIME ETHER COMPOUND AND PHARMACEUTICAL COMPOSITION CONTAINING IT KAKEN PHARMACEUTICAL CO., LTD. (JP) 1993-09-29 EP disclosed
US-4971985-A ANTIISCHEMIC AGENTS, CARDIOVASCULAR DISORDERS KAKEN PHARMACEUTICAL CO., LTD. (JP) 1990-11-20 US disclosed
EP-0366006-A1 Pyridylketoxime ether compound and pharmaceutical composition containing it KAKEN PHARMACEUTICAL CO., LTD. (JP) 1990-05-02 EP disclosed