SCHEMBL9535069

SCHEMBL9535069

COC(=O)c1cc(OC)ccc1N(CC#N)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 6/20 0.43
MTNR1B P49286 6/20 0.43
KDM4E B2RXH2 4/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
HSD17B10 Q99714 3/20 0.41
ALDH1A1 P00352 3/20 0.41
NPC1 O15118 2/20 0.41
LMNA P02545 2/20 0.41
MAPT P10636 2/20 0.41
HPGD P15428 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
TP53 P04637 1/20 0.41
ALOX12 P18054 1/20 0.41
PLA2G2A P14555 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9536183 0.90 MTNR1A (0.43) MTNR1AMTNR1BKDM4EHSD17B10ALDH1A1
SCHEMBL10654450 0.83 MTNR1A (0.44) MTNR1AMTNR1BKDM4ECYP1A2CYP2D6
SCHEMBL24708884 0.74 MTNR1B (0.53) MTNR1AMTNR1B
SCHEMBL341538 0.74 KEAP1 (0.47) MTNR1AMTNR1BKDM4ESMN1; SMN2POLB
SCHEMBL3122141 0.73 KDM4E (0.46) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL21676556 0.72 KDM4E (0.51) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL17659280 0.71 PLA2G2A (0.47) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL3426911 0.69 MTNR1B (0.49) MTNR1AMTNR1BALDH1A1TP53
SCHEMBL14770852 0.68 KMT2A (0.51) KDM4EHSD17B10ALDH1A1LMNAMAPT
SCHEMBL7021315 0.68 KMT2A (0.51) KDM4EHSD17B10ALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0186367-B1 ACIDIC INDOLE COMPOUNDS AND THEIR USE AS ANTIALLERGY AGENTS WARNER-LAMBERT COMPANY (US) 1993-03-03 EP disclosed
US-4675332-A Acidic tetrazolyl substituted indole compounds and their use as antiallergy agents WARNER-LAMBERT COMPANY (US) 1987-06-23 US disclosed
EP-0186367-A2 Acidic indole compounds and their use as antiallergy agents WARNER-LAMBERT COMPANY (US) 1986-07-02 EP disclosed