SCHEMBL9537122

SCHEMBL9537122

COc1cc(Cc2ccc(F)cc2)c(N)c(N)n1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.43
MPO P05164 2/20 0.41
ADCY10 Q96PN6 1/20 0.39
BACE1 P56817 1/20 0.39
HTT P42858 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP2D6 P10635 1/20 0.38
ATM Q13315 1/20 0.38
GRM2 Q14416 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
GPR55 Q9Y2T6 1/20 0.36
LTA4H P09960 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL57463 0.80 MPO (0.56) MPOADCY10
SCHEMBL28488593 0.74 P2RX3 (0.39) DHFRHTTALDH1A1
SCHEMBL28960523 0.71 MPO (0.45) MPOADCY10ALDH1A1
SCHEMBL9536859 0.71 ADORA2A (0.46) MPOALDH1A1CNR1CNR2
SCHEMBL9536206 0.71 TXNRD1 (0.37) DHFRHTTALDH1A1
SCHEMBL28965174 0.71 MAPT (0.42) MPOADCY10ALDH1A1CNR1CNR2
SCHEMBL2419053 0.70 KDM4E (0.49) MPOALDH1A1CYP2D6ATM
SCHEMBL28960530 0.69 LMNA (0.44) DHFRMPOADCY10HTTCNR2
SCHEMBL3844233 0.69 NPC1 (0.32) DHFRALDH1A1
SCHEMBL9538832 0.69 GAA (0.43) DHFRHTTALDH1A1GPR55LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed
EP-0151826-A1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1985-08-21 EP disclosed