SCHEMBL9537232

SCHEMBL9537232

CCC(=C(C(=O)O)C(=O)O)N(CC)c1ccc(F)c(F)c1O

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.33
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
EPHX2 P34913 1/20 0.30
RIPK1 Q13546 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8622658 0.88 EPHX2 (0.36) TSHRALDH1A1GLAEPHX2RIPK1
SCHEMBL1345003 0.73 ALDH1A1 (0.36) TSHRALDH1A1GLARIPK1
SCHEMBL2487489 0.70 TSHR (0.36) TSHRALDH1A1GLA
SCHEMBL17769749 0.70 TSHR (0.43) TSHRALDH1A1
SCHEMBL8621817 0.66 ALDH1A1 (0.30) TSHRALDH1A1GLA
SCHEMBL14845241 0.66 CES2 (0.50) RIPK1
SCHEMBL2475462 0.65 ALDH1A1 (0.44) TSHRALDH1A1GLA
Propionic Acid SCHEMBL29009760 0.64 CES2 (0.50) TSHRALDH1A1EPHX2RIPK1
SCHEMBL9128725 0.63 MAPT (0.32) TSHRALDH1A1EPHX2
SCHEMBL1261683 0.63 HSP90AB1 (0.47) TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0259804-B1 Pyrido[3,2,1-ij]-1,3,4-benzoxadiazine derivatives, process for their preparation, resulting pharmaceutical preparations and intermediates for use in the process HOFFMANN LA ROCHE (CH) 1993-11-18 EP disclosed
EP-0259804-A2 Pyrido[3,2,1-ij]-1,3,4-benzoxadiazine derivatives, process for their preparation, resulting pharmaceutical preparations and intermediates for use in the process F. HOFFMANN-LA ROCHE AG (CH) 1988-03-16 EP disclosed