SCHEMBL8622658

SCHEMBL8622658

CCC(=C(C(=O)O)C(=O)O)N(CC)c1ccc(F)c(F)c1F

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.36
TSHR P16473 2/20 0.34
ALDH1A1 P00352 2/20 0.34
GLA P06280 1/20 0.34
RIPK1 Q13546 1/20 0.34
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
ALPL P05186 1/20 0.30
ALPI P09923 1/20 0.30
ALPG P10696 1/20 0.30
LMNA P02545 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9537232 0.88 TSHR (0.33) EPHX2TSHRALDH1A1GLARIPK1
SCHEMBL1345003 0.75 ALDH1A1 (0.36) TSHRALDH1A1GLARIPK1CES2
SCHEMBL9128725 0.73 MAPT (0.32) EPHX2TSHRALDH1A1LMNA
SCHEMBL2487489 0.72 TSHR (0.36) TSHRALDH1A1GLA
SCHEMBL17769749 0.72 TSHR (0.43) TSHRALDH1A1SMN1; SMN2
SCHEMBL2334592 0.71 EPHX2 (0.38) EPHX2ALDH1A1RIPK1CES2CES1
SCHEMBL14845241 0.71 CES2 (0.50) RIPK1CES2CES1ALPLALPI
Propionic Acid SCHEMBL29009760 0.70 CES2 (0.50) EPHX2TSHRALDH1A1RIPK1CES2
SCHEMBL8621652 0.70 EPHX2 (0.35) EPHX2ALDH1A1RIPK1CES2CES1
SCHEMBL20550632 0.68 TSHR (0.42) TSHRALDH1A1GLARIPK1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0684942-B1 METHOD FOR PREPARING QUINOLINE CARBOXYLIC ACIDS AND DERIVATIVES THEREOF HOECHST CELANESE CORP (US) 1998-06-10 EP disclosed
US-5430152-A Heating aminoarylester in presence of chlorosulfonic acid, oleum HOECHST CELANESE CORPORATION (US) 1995-07-04 US disclosed