SCHEMBL9537277

SCHEMBL9537277

COc1c(Cl)cc(N)c(N)c1Cc1ccc(F)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
GPR55 Q9Y2T6 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
BACE1 P56817 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
ALDH1A1 P00352 5/20 0.35
GAA P10253 2/20 0.35
POLB P06746 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
CYP3A4 P08684 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
CYP2D6 P10635 1/20 0.34
ATM Q13315 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.33
MAOB P27338 1/20 0.33
ADCY10 Q96PN6 1/20 0.33
AR P10275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535642 0.84 SMN1; SMN2 (0.43) CNR1CNR2GPR55L3MBTL1ALDH1A1
SCHEMBL9536290 0.80 GAA (0.41) BACE1NPSR1ALDH1A1GAAPOLB
SCHEMBL9538789 0.73 ALDH1A1 (0.46) L3MBTL1ALDH1A1GAAPOLBHPGD
SCHEMBL9535895 0.70 CNR1 (0.41) CNR1CNR2GPR55ALDH1A1GAA
SCHEMBL9536285 0.67 SLC2A1 (0.38) ALDH1A1GAAHPGDLMNAMAPT
SCHEMBL28412705 0.67 GAA (0.47) ALDH1A1GAAHPGDCYP3A4
SCHEMBL17633590 0.67 CSNK2A1 (0.43) CNR1CNR2L3MBTL1NPSR1ALDH1A1
SCHEMBL22588510 0.66 GAA (0.41) ALDH1A1GAAHPGD
SCHEMBL29449610 0.66 GAA (0.41) ALDH1A1GAAHPGD
SCHEMBL8892263 0.65 THRB (0.43) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed
EP-0151826-A1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1985-08-21 EP disclosed