SCHEMBL9537470

SCHEMBL9537470

OCCN1CCC(Cc2nc3ccccc3n2Cc2ccco2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.50
HRH1 P35367 4/20 0.48
TSHR P16473 2/20 0.47
POLB P06746 2/20 0.47
ALDH1A1 P00352 2/20 0.47
USP2 O75604 1/20 0.47
HSD17B10 Q99714 1/20 0.47
ATM Q13315 1/20 0.41
CYP2D6 P10635 1/20 0.41
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40
DRD3 P35462 1/20 0.40
GRM2 Q14416 1/20 0.40
GAA P10253 1/20 0.40
TRPC4 Q9UBN4 1/20 0.39
TRPC5 Q9UL62 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535315 0.90 ALDH1A1 (0.47) KDM4ETSHRPOLBALDH1A1USP2
SCHEMBL9537714 0.87 ALDH1A1 (0.45) KDM4ETSHRALDH1A1USP2HSD17B10
SCHEMBL9539854 0.87 ALDH1A1 (0.52) KDM4EHRH1TSHRALDH1A1USP2
SCHEMBL9535911 0.85 ALDH1A1 (0.43) KDM4ETSHRALDH1A1USP2HSD17B10
SCHEMBL9535187 0.85 ALDH1A1 (0.45) KDM4ETSHRPOLBALDH1A1USP2
SCHEMBL9536425 0.85 KDM4E (0.43) KDM4EHRH1TSHRPOLBALDH1A1
Fumaric Acid SCHEMBL11069587 0.84 ALDH1A1 (0.41) KDM4EHRH1TSHRPOLBALDH1A1
SCHEMBL9536155 0.84 USP2 (0.42) KDM4EHRH1TSHRPOLBALDH1A1
SCHEMBL9537584 0.84 MEN1 (0.56) KDM4EHRH1TSHRPOLBALDH1A1
SCHEMBL9535185 0.84 MAPT (0.49) KDM4EPOLBALDH1A1USP2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed
US-4839374-A TREATING ALLERGIES JANSSEN PHARMACEUTICA, N.V. (BE) 1989-06-13 US disclosed
US-4695575-A ANTIHISTAMINES JANSSEN PHARMACEUTICA, N.V. (BE) 1987-09-22 US disclosed