SCHEMBL9537962

SCHEMBL9537962

COc1ccc(CCN2CCC(Cc3nc4ncccc4n3Cc3ccc(F)cc3)CC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.57
SLC6A4 P31645 4/20 0.57
HRH1 P35367 3/20 0.57
TACR2 P21452 2/20 0.57
TACR1 P25103 2/20 0.57
EED O75530 2/20 0.57
SSTR5 P35346 2/20 0.57
KCNH2 Q12809 2/20 0.57
MEN1 O00255 1/20 0.57
MLNR O43193 1/20 0.57
CACNA1F O60840 1/20 0.57
USP2 O75604 1/20 0.57
ABCB11 O95342 1/20 0.57
EGFR P00533 1/20 0.57
LMNA P02545 1/20 0.57
HLA-A P04439 1/20 0.57
ERBB2 P04626 1/20 0.57
TP53 P04637 1/20 0.57
CYP1A2 P05177 1/20 0.57
LCK P06239 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL10546958 0.95 HRH1 (0.57) HTR1ASLC6A4HRH1TACR2TACR1
SCHEMBL9540175 0.88 KCNH2 (0.71) HTR1ASLC6A4HRH1TACR2TACR1
SCHEMBL9537190 0.84 PRMT3 (0.44) HRH1SSTR5KCNH2CYP2D6CHRM1
SCHEMBL10547773 0.83 HTR1A (0.56) HTR1ASLC6A4HRH1TACR2TACR1
SCHEMBL1151559 0.83 KCNH2 (0.78) HTR1ASLC6A4HRH1TACR2TACR1
Hydrochloric Acid SCHEMBL9537185 0.82 HTR1A (0.57) HTR1ASLC6A4HRH1TACR2TACR1
SCHEMBL9536547 0.82 SSTR5 (0.52) SLC6A4SSTR5HTR3ASLC6A3
SCHEMBL9564828 0.82 HRH1 (0.49) HTR1ASLC6A4HRH1TACR2TACR1
SCHEMBL9696669 0.82 HRH1 (0.55) HTR1ASLC6A4HRH1TACR2TACR1
SCHEMBL9537882 0.81 SLC6A9 (0.41) HTR1AHRH1SSTR5KCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed