SCHEMBL9540217

SCHEMBL9540217

NCCN1CCN(C(F)(F)F)CC1c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.40
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA7 P36544 1/20 0.34
CHRNA4 P43681 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
NR1H2 P55055 10/20 0.34
NR1H3 Q13133 9/20 0.34
MAPK1 P28482 1/20 0.34
PRMT3 O60678 1/20 0.33
CARM1 Q86X55 1/20 0.33
PRMT6 Q96LA8 1/20 0.33
PRMT1 Q99873 1/20 0.33
PRMT8 Q9NR22 1/20 0.33
RIPK1 Q13546 1/20 0.33
KIF11 P52732 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8057149 0.83 P2RX7 (0.41) P2RX7CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL18824255 0.79 MAPK1 (0.46) P2RX7CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL10927522 0.79 P2RX7 (0.37) P2RX7NR1H2NR1H3
Hydrochloric Acid SCHEMBL3670802 0.78 SIGMAR1 (0.44) P2RX7PRMT3CARM1PRMT6PRMT1
Hydrochloric Acid SCHEMBL3670800 0.74 P2RX7 (0.41) P2RX7CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL9199829 0.74 SIGMAR1 (0.40) P2RX7CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL11452553 0.72 CHRNB2 (0.56) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL506196 0.71 RECQL (0.45) PRMT3CARM1PRMT6PRMT1PRMT8
SCHEMBL4714894 0.71 CHRNB2 (0.50) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL25533005 0.70 P2RX7 (0.54) P2RX7CHRNB2CHRNB4CHRNA3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993003016-A1 BENZIMIDAZOLONE DERIVATIVES AS 5-HT1A AND 5-HT2 ANTAGONISTS BOEHRINGER INGELHEIM ITALIA S.P.A. (IT) 1993-02-18 WO disclosed