SCHEMBL8057149

SCHEMBL8057149

FC(F)(F)N1CCN(CCCCl)C(c2ccccc2)C1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.41
NR1H2 P55055 15/20 0.34
NR1H3 Q13133 15/20 0.34
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA7 P36544 1/20 0.33
CHRNA4 P43681 1/20 0.33
PHGDH O43175 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9540217 0.83 P2RX7 (0.40) P2RX7NR1H2NR1H3CHRNB2CHRNB4
SCHEMBL10927522 0.77 P2RX7 (0.37) P2RX7NR1H2NR1H3
SCHEMBL11860669 0.73 CHRNB2 (0.47) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL27820682 0.69 CHRNB2 (0.40) P2RX7CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL9199829 0.69 SIGMAR1 (0.40) P2RX7CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL25533005 0.68 P2RX7 (0.54) P2RX7NR1H2NR1H3CHRNB2CHRNB4
SCHEMBL11938944 0.67 MAPK1 (0.42) P2RX7
SCHEMBL11932483 0.65 HSP90AA1 (0.41) P2RX7CHRNB2CHRNB4CHRNA3CHRNA7
Hydrochloric Acid SCHEMBL3672966 0.65 SIGMAR1 (0.49)
SCHEMBL27979543 0.63 DRD2 (0.42) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998923-A1 Use of 5-HT7 receptor agonists for the treatment or prophylaxis of ischemias BASF AKTIENGESELLSCHAFT (DE) 2000-05-10 EP disclosed