SCHEMBL9540318

SCHEMBL9540318

O=c1cc[nH]c(=O)n1CCN1CCC(Cc2nc3ccccc3n2Cc2ccco2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.41
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 2/20 0.41
USP2 O75604 2/20 0.41
HSD17B10 Q99714 2/20 0.41
NOS2 P35228 3/20 0.39
NOS3 P29474 2/20 0.39
NOS1 P29475 2/20 0.39
ATM Q13315 1/20 0.38
MAPT P10636 2/20 0.37
MAPK1 P28482 3/20 0.37
NPSR1 Q6W5P4 2/20 0.37
GAA P10253 2/20 0.37
CFTR P13569 1/20 0.37
HRH1 P35367 1/20 0.37
TDP1 Q9NUW8 2/20 0.36
HTT P42858 1/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9537087 0.83 TSHR (0.54) TSHRALDH1A1MAPTMAPK1NPSR1
SCHEMBL9537470 0.82 KDM4E (0.50) TSHRALDH1A1KDM4EUSP2HSD17B10
SCHEMBL9535315 0.82 ALDH1A1 (0.47) TSHRALDH1A1KDM4EUSP2HSD17B10
SCHEMBL9538853 0.81 P2RX7 (0.49) USP2MAPK1HRH1MEN1KMT2A
Hydrochloric Acid SCHEMBL9537429 0.81 GAA (0.52) TSHRALDH1A1KDM4EUSP2HSD17B10
SCHEMBL9539277 0.80 ALDH1A1 (0.49) TSHRALDH1A1KDM4EHSD17B10MAPT
SCHEMBL9537714 0.80 ALDH1A1 (0.45) TSHRALDH1A1KDM4EUSP2HSD17B10
SCHEMBL9539854 0.80 ALDH1A1 (0.52) TSHRALDH1A1KDM4EUSP2HSD17B10
SCHEMBL10551946 0.79 TSHR (0.52) TSHRALDH1A1HSD17B10MAPTMAPK1
SCHEMBL9535911 0.79 ALDH1A1 (0.43) TSHRALDH1A1KDM4EUSP2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP claimed