SCHEMBL9537087

SCHEMBL9537087

O=c1[nH]c2ccccc2c(=O)n1CCN1CCC(Cc2nc3ccccc3n2Cc2ccco2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.54
ACHE P22303 1/20 0.48
ALDH1A1 P00352 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
HTR1A P08908 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C9 P11712 1/20 0.44
DRD2 P14416 1/20 0.44
HPGD P15428 1/20 0.44
ADRA2B P18089 1/20 0.44
ADRA2C P18825 1/20 0.44
DRD1 P21728 1/20 0.44
DRD4 P21917 1/20 0.44
HTR1D P28221 1/20 0.44
HTR1B P28222 1/20 0.44
HTR2A P28223 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10551946 0.95 TSHR (0.52) TSHRACHEALDH1A1MEN1KMT2A
SCHEMBL9539277 0.92 ALDH1A1 (0.49) TSHRALDH1A1MEN1KMT2ACYP1A2
SCHEMBL9538853 0.87 P2RX7 (0.49) MEN1KMT2ALMNACYP1A2CYP3A4
SCHEMBL9538362 0.85 ACHE (0.48) TSHRACHEALDH1A1MEN1KMT2A
SCHEMBL10550979 0.85 TSHR (0.50) TSHRACHEALDH1A1MEN1KMT2A
SCHEMBL9540587 0.85 TSHR (0.50) TSHRACHEALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL9537429 0.85 GAA (0.52) TSHRALDH1A1MEN1KMT2ALMNA
SCHEMBL9540318 0.83 TSHR (0.41) TSHRALDH1A1MEN1KMT2AMAPT
SCHEMBL9540183 0.83 ACHE (0.47) TSHRACHEALDH1A1MEN1KMT2A
SCHEMBL9539651 0.82 ALDH1A1 (0.47) TSHRALDH1A1KMT2ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP claimed