SCHEMBL9564149

SCHEMBL9564149

Cn1cc(Cc2ccc(C(=O)OC(C)(C)C)cc2)c2c(O)nc(N)nc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
HSP90AA1 P07900 4/20 0.34
DHFR P00374 2/20 0.34
SIRT2 Q8IXJ6 1/20 0.34
SIRT1 Q96EB6 1/20 0.34
ADCY10 Q96PN6 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
THRB P10828 1/20 0.32
HPGD P15428 1/20 0.32
HIF1A Q16665 1/20 0.32
SMO Q99835 1/20 0.32
SLC7A5 Q01650 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564205 0.78 TYMS (0.43) DHFR
SCHEMBL9844768 0.74 TBXAS1 (0.39) ALDH1A1MAPT
SCHEMBL9564148 0.73 L3MBTL1 (0.45) DHFRKDM4EALDH1A1HPGD
SCHEMBL9564146 0.73 L3MBTL1 (0.45) DHFRKDM4EALDH1A1HPGD
SCHEMBL7653891 0.70 CA12 (0.43) CA12CA1CA2CA9CA14
SCHEMBL7708759 0.69 KMT2A (0.52) CA12CA1CA2CA9CA14
SCHEMBL9001785 0.67 TLR7 (0.44) CA12CA1CA2CA9CA14
SCHEMBL9446061 0.66 TLR8 (0.39) DHFRSLC7A5TLR8TLR7
SCHEMBL12918481 0.66 CDK1 (0.33)
SCHEMBL422913 0.64 LOXL2 (0.65) CA12CA1CA2CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0549291-A1 Thymidylate synthase inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-06-30 EP disclosed