SCHEMBL9566833

SCHEMBL9566833

O=C(Nc1ccc(F)cc1)c1ccc(CO)nc1

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
P4HTM Q9NXG6 2/20 0.63
CXCR2 P25025 10/20 0.59
CXCR1 P25024 7/20 0.57
PTPN1 P18031 2/20 0.56
PTPN6 P29350 1/20 0.56
PTPN11 Q06124 1/20 0.56
KCNQ3 O43525 1/20 0.55
KCNQ2 O43526 1/20 0.55
KCNE1 P15382 1/20 0.55
KCNQ1 P51787 1/20 0.55
BACE1 P56817 1/20 0.55
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
KMT2A Q03164 1/20 0.54
ALDH1A1 P00352 1/20 0.54
MITF O75030 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9566852 0.92 P4HTM (0.55) P4HTMCXCR2CXCR1PTPN1PTPN6
SCHEMBL9517015 0.89 P4HTM (0.51) P4HTMCXCR2CXCR1PTPN1PTPN6
SCHEMBL9566835 0.85 P4HTM (0.63) P4HTMKCNQ3KCNQ2KCNE1KCNQ1
SCHEMBL9566802 0.85 NPC1 (0.67) P4HTMCXCR2CXCR1PTPN1KMT2A
SCHEMBL9566902 0.83 CXCR2 (0.62) P4HTMCXCR2CXCR1PTPN1PTPN6
SCHEMBL9566803 0.82 P4HTM (0.66) P4HTMCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL9566776 0.82 P4HTM (0.66) P4HTMCXCR2CXCR1KMT2AALDH1A1
SCHEMBL9566786 0.81 CXCR2 (0.57) P4HTMCXCR2CXCR1ALDH1A1
SCHEMBL9566868 0.81 CXCR2 (0.60) P4HTMCXCR2CXCR1ALDH1A1
SCHEMBL9566887 0.81 P4HTM (0.69) P4HTMCYP1A2CYP3A4KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0533130-A1 2-Hydroxymethylpyridines, the corresponding pyridine-N-oxides and derivatives thereof, process for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1993-03-24 EP disclosed