SCHEMBL9568317

SCHEMBL9568317

COc1c(-c2ccc(CN)cc2)c(F)cc2c(=O)c(C(=O)O)c3n(c12)C(c1ccc(F)cc1F)S3

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 9/20 0.40
NR1H2 P55055 6/20 0.34
NR1H3 Q13133 6/20 0.34
NEK1 Q96PY6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9568311 0.92 TOP1 (0.41) TOP1NR1H2NR1H3NEK1
SCHEMBL9568346 0.89 TOP1 (0.40) TOP1NEK1
SCHEMBL9568432 0.87 TOP1 (0.39) TOP1NEK1
SCHEMBL9568467 0.80 GSK3B (0.36) TOP1
SCHEMBL9568342 0.80 TOP1 (0.34) TOP1
SCHEMBL9568385 0.79 LMNA (0.35) TOP1
SCHEMBL9568333 0.79 TOP1 (0.39) TOP1NEK1
Hydrochloric Acid SCHEMBL9568570 0.78 LMNA (0.36) TOP1
SCHEMBL9568460 0.78 TOP2A (0.39) TOP1NEK1
SCHEMBL9568358 0.78 PRKCZ (0.37) TOP1NEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0551518-A1 QUINOLINECARBOXYLIC ACID DERIVATIVE NIPPON SHINYAKU COMPANY, LIMITED (JP) 1993-07-21 EP disclosed