SCHEMBL9568520

SCHEMBL9568520

N=C(N)c1ccc(-c2ccc(-n3cnc(CC(N)C(=O)O)c3)nn2)cc1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 2/20 0.36
CPB2 Q96IY4 6/20 0.36
CPB1 P15086 5/20 0.36
CYP1A2 P05177 1/20 0.34
MAP4K4 O95819 1/20 0.33
F10 P00742 3/20 0.32
CPN1 P15169 1/20 0.32
F9 P00740 1/20 0.32
TPH1 P17752 2/20 0.32
ITGB3 P05106 1/20 0.32
ITGA2B P08514 1/20 0.32
F2 P00734 1/20 0.31
PRSS1 P07477 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9256051 0.99 PDK1 (0.36) PDK1CPB2CPB1CYP1A2MAP4K4
SCHEMBL9254878 0.90 CPB2 (0.36) PDK1CPB2CPB1MAP4K4F10
SCHEMBL9258718 0.89 CPB1 (0.39) PDK1CPB2CPB1F10F9
SCHEMBL9568746 0.88 F10 (0.36) PDK1CPB2CPB1F10ITGB3
SCHEMBL9248830 0.87 CPB2 (0.42) PDK1CPB2CPB1F10F9
SCHEMBL9251486 0.86 ITGB3 (0.36) PDK1CPB2CPB1MAP4K4F10
SCHEMBL9255144 0.86 TPH1 (0.39) CPB2CPB1MAP4K4TPH1
SCHEMBL9568572 0.85 PDK1 (0.39) PDK1CPB2CPB1CYP1A2TPH1
Trifluoroacetic Acid SCHEMBL9095103 0.85 F10 (0.36) CPB2CPB1F10F9ITGB3
Hydrochloric Acid SCHEMBL9255416 0.84 PDK1 (0.39) PDK1CPB2CPB1CYP1A2TPH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP claimed