SCHEMBL9569693

SCHEMBL9569693

FC(F)(F)C1=NC(C(F)(F)F)Cc2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 11/20 0.38
NOS2 P35228 9/20 0.38
PNMT P11086 1/20 0.35
ACHE P22303 1/20 0.33
CYP19A1 P11511 1/20 0.31
TSHR P16473 1/20 0.31
HTR2A P28223 1/20 0.31
NOS1 P29475 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3248266 0.79 NOS3 (0.38) NOS3NOS2PNMTACHECYP19A1
SCHEMBL638089 0.79 NOS3 (0.41) NOS3NOS2PNMTACHECYP19A1
SCHEMBL637334 0.76 NOS3 (0.35) NOS3NOS2PNMTACHECYP19A1
SCHEMBL7298902 0.66 NOS3 (0.53) NOS3NOS2CYP19A1TSHRHTR2A
SCHEMBL29964099 0.66 NOS3 (0.53) NOS3NOS2CYP19A1TSHRHTR2A
SCHEMBL7310501 0.64 PNMT (0.37) PNMTCYP19A1
Hydrochloric Acid SCHEMBL11781894 0.63 PNMT (0.36) NOS2PNMTHTR2ANOS1
SCHEMBL11523523 0.62 ACHE (0.53) PNMTACHECYP19A1TSHR
SCHEMBL28529344 0.62 HTR2A (0.49) NOS3NOS2PNMTACHETSHR
SCHEMBL29407071 0.62 HTR2A (0.49) NOS3NOS2PNMTACHETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5204471-A α-trifluoromethyl-substituted, saturated bicyclic amines BAYER AKTIENGESELLSCHAFT (DE) 1993-04-20 US disclosed
EP-0527385-A1 Alpha-trifluoromethyl substituted, saturated bicyclic amines and process for their preparation BAYER AG (DE) 1993-02-17 EP disclosed