SCHEMBL9575341

SCHEMBL9575341

C=C(F)C(=O)Oc1ccc(C)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.42
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
ACHE P22303 2/20 0.38
NPC1 O15118 3/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
KMT2A Q03164 2/20 0.35
RAB9A P51151 3/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PRNP P04156 1/20 0.34
GAA P10253 1/20 0.34
ELANE P08246 1/20 0.34
KMO O15229 2/20 0.33
SLC6A3 Q01959 1/20 0.33
MAPT P10636 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9575371 0.87 CHEK2 (0.37) ACHENPC1L3MBTL1TDP1KMT2A
SCHEMBL20344359 0.87 ELANE (0.47) MRGPRX4HDAC1HDAC6ACHENPC1
SCHEMBL12636049 0.84 CES2 (0.39) NPC1KMT2ARAB9AGAAELANE
SCHEMBL17355789 0.81 HDAC1 (0.45) MRGPRX4HDAC1HDAC6ACHENPC1
SCHEMBL1432110 0.79 ACHE (0.59) MRGPRX4HDAC1HDAC6ACHETDP1
SCHEMBL18869516 0.78 THRB (0.46) MRGPRX4HDAC1HDAC6ACHENPC1
SCHEMBL3879835 0.77 MRGPRX4 (0.44) MRGPRX4HDAC1HDAC6ACHENPC1
SCHEMBL27565314 0.77 KMT2A (0.52) MRGPRX4HDAC1HDAC6ACHENPC1
SCHEMBL9575396 0.77 LMNA (0.55) L3MBTL1KMT2AALDH1A1GAAELANE
SCHEMBL9575641 0.77 MAPT (0.42) NPC1KMT2ARAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5266668-A Substituted phenyl α-fluoroacrylates HOECHST AKTIENGESELLSCHAFT (DE) 1993-11-30 US disclosed
EP-0249867-B1 SUBSTITUTED PHENYL ESTERS OF ALPHA-FLUOROACRYLIC ACID HOECHST AKTIENGESELLSCHAFT (DE) 1992-01-02 EP disclosed
EP-0249867-A2 Substituted phenyl esters of alpha-fluoroacrylic acid HOECHST AKTIENGESELLSCHAFT (DE) 1987-12-23 EP disclosed