SCHEMBL9575441

SCHEMBL9575441

CC(=O)Nc1ncc2ncn(COC(CCOC(C)C)OCc3ccccc3)c2n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KA3 P51812 1/20 0.35
BRD4 O60885 1/20 0.35
ALDH1A1 P00352 4/20 0.35
HPGD P15428 2/20 0.35
HSD17B10 Q99714 2/20 0.35
KDM4E B2RXH2 2/20 0.35
ADRA1A P35348 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
TSHR P16473 3/20 0.33
CYP1A2 P05177 2/20 0.33
CLK4 Q9HAZ1 1/20 0.33
JAK3 P52333 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA1 P30542 1/20 0.32
ACHE P22303 2/20 0.32
APP P05067 1/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9575565 0.87 RPS6KA3 (0.39) RPS6KA3ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL9575536 0.85 ACHE (0.43) BRD4TSHRACHE
SCHEMBL9575800 0.85 ALDH1A1 (0.40) ALDH1A1HPGDHSD17B10KDM4EADRA1A
SCHEMBL9575434 0.84 CYP1A2 (0.37) RPS6KA3BRD4ALDH1A1HPGDHSD17B10
SCHEMBL9575559 0.79 ALDH1A1 (0.41) RPS6KA3ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL9575560 0.71 ACHE (0.40) ALDH1A1TSHRACHECYP3A4HIF1A
SCHEMBL9019800 0.71 BCHE (0.38) BRD4HPGDTSHRCYP1A2ACHE
SCHEMBL9845246 0.71 BCHE (0.36) BRD4HPGDTSHRCYP1A2ACHE
SCHEMBL9575400 0.70 KDM4E (0.46) RPS6KA3ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL10816876 0.70 PDE3A (0.38) ALDH1A1HPGDHSD17B10KDM4EADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5225550-A PROCESS FOR THE PREPARATION OF SUBSTITUTED ACYCLIC NUCLEOSIDES, AND INTERMEDIATES OCCURRING THEREIN HOECHST AKTIENGESELLSCHAFT (DE) 1993-07-06 US disclosed
CN-1057652-A A kind of acyclic nucleotide of replacement and method of related intermediates thereof of preparing HOECHST AG (DE) 1992-01-08 CN disclosed