SCHEMBL9587666

SCHEMBL9587666

CC1(C)C=C(n2ccccc2=O)c2cc(C#C[Si](C)(C)C)ccc2C1=O

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.37
GABRG2 P18507 2/20 0.37
GABRB3 P28472 2/20 0.37
GABRA5 P31644 2/20 0.37
GABRA3 P34903 2/20 0.37
GABRA2 P47869 2/20 0.37
ABCC9 O60706 1/20 0.35
ABCC8 Q09428 1/20 0.35
KCNJ11 Q14654 1/20 0.35
KCNJ8 Q15842 1/20 0.35
ADK P55263 2/20 0.33
GRM5 P41594 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6369766 0.84 ABCC9 (0.50) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL9587437 0.84 ABCC9 (0.38) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL9587196 0.79 ABCC9 (0.47) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL9587001 0.77 CA1 (0.39) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9589242 0.77 CA1 (0.39) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9587407 0.77 S100A4 (0.36)
SCHEMBL9590341 0.75 GFER (0.36)
SCHEMBL9589861 0.75 ALDH1A1 (0.42)
SCHEMBL9590296 0.75 CA1 (0.43)
SCHEMBL9587505 0.74 SLC6A9 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5208246-A Hypotensive, bronchodilator J. URIACH & CIA. (ES) 1993-05-04 US claimed
EP-0489300-A2 Tetralones with pharmacological activity J. URIACH & CIA. S.A. (ES) 1992-06-10 EP claimed
US-5272170-A Tetralones with pharmacological activity J. URIACH & CIA., S.A. (ES) 1993-12-21 US disclosed
US-5208246-A Hypotensive, bronchodilator J. URIACH & CIA. (ES) 1993-05-04 US disclosed
EP-0489300-A2 Tetralones with pharmacological activity J. URIACH & CIA. S.A. (ES) 1992-06-10 EP disclosed