SCHEMBL9587196

SCHEMBL9587196

CC1(C)C=C(n2ccccc2=O)c2ccc(C#N)cc2C1=O

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 2/20 0.47
ABCC8 Q09428 1/20 0.47
KCNJ11 Q14654 1/20 0.47
KCNJ8 Q15842 1/20 0.47
PGR P06401 2/20 0.35
CASP3 P42574 1/20 0.35
HTR1A P08908 4/20 0.34
F10 P00742 1/20 0.34
MALT1 Q9UDY8 1/20 0.33
GABRA1 P14867 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32
GABRA3 P34903 1/20 0.32
GABRA2 P47869 1/20 0.32
NSD2 O96028 1/20 0.32
G6PD P11413 2/20 0.32
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6369766 0.95 ABCC9 (0.50) ABCC9ABCC8KCNJ11KCNJ8PGR
SCHEMBL9587437 0.83 ABCC9 (0.38) ABCC9ABCC8KCNJ11KCNJ8GABRA1
SCHEMBL9588407 0.81 CA1 (0.39) F10CA1CA2
SCHEMBL9589614 0.80 ABCC9 (0.38) ABCC9ABCC8KCNJ11KCNJ8PGR
SCHEMBL9587666 0.79 GABRA1 (0.37) ABCC9ABCC8KCNJ11KCNJ8GABRA1
SCHEMBL9733561 0.79 PGR (0.36) ABCC9ABCC8KCNJ11KCNJ8PGR
Bimakalim SCHEMBL231904 0.79 PDE4A (0.43) ABCC9ABCC8KCNJ11KCNJ8CASP3
SCHEMBL9733284 0.79 HTR1A (0.37) ABCC9ABCC8KCNJ11KCNJ8PGR
SCHEMBL8088443 0.79 MAOB (0.38) ABCC9ABCC8KCNJ11KCNJ8PGR
SCHEMBL9587505 0.78 SLC6A9 (0.33) PGRF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5272170-A Tetralones with pharmacological activity J. URIACH & CIA., S.A. (ES) 1993-12-21 US disclosed
US-5208246-A Hypotensive, bronchodilator J. URIACH & CIA. (ES) 1993-05-04 US disclosed
EP-0489300-A2 Tetralones with pharmacological activity J. URIACH & CIA. S.A. (ES) 1992-06-10 EP disclosed