SCHEMBL9596069

SCHEMBL9596069

CCOC(=O)[C@H](CC(C)C)NS(=O)(=O)c1ccc(S(=O)(=O)c2ccccc2)s1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
CYP2C9 P11712 2/20 0.41
CTSL P07711 3/20 0.41
CTSS P25774 3/20 0.41
CTSK P43235 3/20 0.41
TSHR P16473 1/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
MAPT P10636 3/20 0.40
LARS1 Q9P2J5 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP2C19 P33261 1/20 0.39
MMP1 P03956 1/20 0.39
MMP2 P08253 1/20 0.39
MMP3 P08254 1/20 0.39
MMP7 P09237 1/20 0.39
MMP9 P14780 1/20 0.39
MMP13 P45452 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7061397 0.87 MMP2 (0.51) KMT2AMEN1CYP2C9CTSLCTSS
SCHEMBL9596098 0.74 TDP1 (0.54) BACE1KMT2AMEN1CYP2C9ALDH1A1
SCHEMBL7060922 0.73 MMP2 (0.48) KMT2AMEN1CYP2C9CTSLCTSS
SCHEMBL24855401 0.72 CTSK (0.57) CTSLCTSSCTSKMMP1MMP2
SCHEMBL18775046 0.72 CTSK (0.57) CTSLCTSSCTSKMMP1MMP2
SCHEMBL6795703 0.72 CTSL (0.53) BACE1KMT2AMEN1CTSLCTSS
SCHEMBL9596076 0.72 ALDH1A1 (0.46) KMT2AMEN1CYP2C9TSHRMAPT
SCHEMBL16388801 0.71 CTSL (0.57) CTSLCTSSCTSKLARS1MMP1
SCHEMBL8998137 0.71 BACE1 (0.50) BACE1KMT2AMEN1CTSLCTSS
SCHEMBL8133560 0.71 MMP1 (0.51) BACE1KMT2AMEN1CYP2C9CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993015047-A1 AMINO ACID DERIVATIVES AS PAF ANTAGONISTS BRITISH BIO-TECHNOLOGY LIMITED (GB) 1993-08-05 WO claimed
WO-1993015047-A1 AMINO ACID DERIVATIVES AS PAF ANTAGONISTS BRITISH BIO-TECHNOLOGY LIMITED (GB) 1993-08-05 WO disclosed
WO-1993006092-A1 PIPERAZINYL (SULFONYL)AMIDE DERIVATIVES OF CAMPHOR AS OXYTOCIN ANTAGONISTS MERCK & CO., INC. (US) 1993-04-01 WO disclosed