SCHEMBL9601104

SCHEMBL9601104

S=C(Cl)OOc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 3/20 0.38
TSHR P16473 1/20 0.38
CA5A P35218 1/20 0.36
CA5B Q9Y2D0 1/20 0.36
CA4 P22748 1/20 0.35
NR1H2 P55055 1/20 0.34
BAX Q07812 1/20 0.34
ALDH1A1 P00352 2/20 0.33
TAAR1 Q96RJ0 1/20 0.33
RECQL P46063 1/20 0.33
SRC P12931 1/20 0.33
ATM Q13315 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ALOX15 P16050 1/20 0.32
KCNA3 P22001 1/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
CA1 P00915 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7954828 0.80 LTA4H (0.41) LTA4HTSHRCA5ACA5BCA4
SCHEMBL2522708 0.80 LTA4H (0.41) LTA4HTSHRCA5ACA5BCA4
SCHEMBL10626679 0.77 ACHE (0.41) TSHRALDH1A1L3MBTL1MEN1MAPT
SCHEMBL6552309 0.77 MAOB (0.39) ALDH1A1RECQLATMMEN1KMT2A
SCHEMBL8104753 0.77 LTA4H (0.35) LTA4HTSHRCA5ACA5BCA4
SCHEMBL4010662 0.76 ALDH1A1 (0.43) LTA4HTSHRCA5ACA5BALDH1A1
SCHEMBL19247 0.75 LTA4H (0.41) LTA4HTSHRCA5ACA5BCA4
Potassium Ion SCHEMBL28444151 0.74 CA12 (0.47) LTA4HTSHRCA5ACA5BCA4
SCHEMBL10628533 0.73 IDO1 (0.45) ALDH1A1
SCHEMBL10653814 0.73 CYP1A1 (0.39) ALDH1A1MEN1MAPTKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-5310759-A None JP disclosed
JP-H05310759-A INTERMEDIATE FOR PREPARATION OF 2-ALKYLTHIOPEN-2-EM-3-CARBOXYLIC ACID ANTIBIOTIC MERCK & CO INC 1993-11-22 JP disclosed
EP-0320497-A1 Substituted 2-thioxopenams, intermediates therefrom and process for preparing substituted 2-thioxopenams and 2-substituted thiopenems MERCK & CO. INC. (US) 1989-06-14 EP disclosed
US-4675317-A PENICILLIN ANTIBIOTICS MERCK & CO., INC. (US) 1987-06-23 US disclosed
US-4610823-A INTERMEDIATES FOR PENEM ANTIBIOTICS MERCK & CO., INC. (US) 1986-09-09 US disclosed
EP-0115308-A2 2-Unsaturated alkylthio-pen-2-em-3-carboxylic acids and process for preparing substituted 2-thioxopenams and 2-substituted thiopenems MERCK & CO. INC. (US) 1984-08-08 EP disclosed