SCHEMBL9602457

SCHEMBL9602457

O=c1[nH]c2ccccc2n1CCCN1CCC(Cc2nc3cncnc3n2Cc2ccc(F)cc2)CC1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 7/20 0.45
CYP3A4 P08684 6/20 0.45
USP2 O75604 6/20 0.45
CYP2C9 P11712 4/20 0.45
CYP2C19 P33261 3/20 0.45
HIF1A Q16665 3/20 0.45
CYP2D6 P10635 2/20 0.45
LMNA P02545 3/20 0.44
MAPK1 P28482 3/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44
HBB P68871 1/20 0.44
P2RX7 Q99572 1/20 0.43
MEN1 O00255 1/20 0.43
SLC22A2 O15244 1/20 0.43
NR1I2 O75469 1/20 0.43
GMNN O75496 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL9565017 0.94 CYP1A2 (0.48) CYP1A2CYP3A4USP2CYP2C9CYP2C19
SCHEMBL9564927 0.87 P2RX7 (0.44) CYP1A2CYP3A4USP2HIF1ACYP2D6
SCHEMBL9601946 0.85 HTR7 (0.44) LMNAP2RX7HTR1ADRD2HTR2A
SCHEMBL10552682 0.83 USP2 (0.47) CYP1A2CYP3A4USP2HIF1ACYP2D6
SCHEMBL10546931 0.83 GRIN1 (0.47) CYP1A2CYP3A4USP2HIF1ACYP2D6
SCHEMBL9564956 0.82 CYP1A2 (0.54) CYP1A2CYP3A4USP2CYP2C9CYP2C19
SCHEMBL9565027 0.81 SSTR5 (0.55) CYP1A2CYP3A4USP2CYP2C9CYP2C19
Fumaric Acid SCHEMBL9565037 0.81 USP2 (0.46) CYP1A2USP2CYP2D6P2RX7HTR1A
SCHEMBL1152886 0.80 LMNA (0.60) CYP1A2CYP3A4USP2HIF1ACYP2D6
SCHEMBL10550233 0.80 ACHE (0.51) CYP1A2CYP3A4CYP2C9CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0206415-B1 (4-PIPERIDINYLMETHYL AND -HETERO)PURINES JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-27 EP disclosed