SCHEMBL9604977

SCHEMBL9604977

CN[C@@H](Cc1c[nH]c(=S)[nH]1)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC22A4 Q9H015 1/20 0.51
KDM3B Q7LBC6 1/20 0.37
ITGB2 P05107 2/20 0.33
ICAM1 P05362 2/20 0.33
ITGAL P20701 2/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
GFER P55789 1/20 0.32
ALOX15 P16050 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31
ACE P12821 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26882134 0.85 SLC22A4 (0.49) SLC22A4KDM3BITGB2ICAM1ITGAL
SCHEMBL26882364 0.81 SLC22A4 (0.46) SLC22A4KMT2ATDP1KDM4EGAA
SCHEMBL9604220 0.79 SLC22A4 (0.55) SLC22A4KDM3BKMT2ATDP1KDM4E
SCHEMBL12800006 0.76 SLC22A4 (0.51) SLC22A4KDM3BKMT2ATDP1KDM4E
SCHEMBL1867165 0.76 SLC22A4 (0.51) SLC22A4KDM3BKMT2ATDP1KDM4E
SCHEMBL175156 0.75 SLC22A4 (0.76) SLC22A4KDM3BKMT2ATDP1GAA
SCHEMBL745229 0.75 SLC22A4 (0.76) SLC22A4KDM3BKMT2ATDP1GAA
SCHEMBL26882423 0.74 SLC22A4 (0.47) SLC22A4KDM3BKMT2ATDP1KDM4E
SCHEMBL151336 0.70 ITGB2 (0.60) ITGB2ICAM1ITGALKMT2AKDM4E
SCHEMBL163397 0.70 ITGB2 (0.60) ITGB2ICAM1ITGALKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023220754-A1 ANTIOXIDANT DERIVATIVE OF HYALURONIC ACID UNIVERSITY OF VERMONT AND STATE AGRICULTURAL COLLEGE (US) 2023-11-16 WO disclosed
EP-2486020-B1 METHOD FOR THE SYNTHESIS OF ERGOTHIONEINE AND THE LIKE TETRAHEDRON (FR) 2017-08-16 EP disclosed
EP-2486019-B1 METHOD FOR THE SYNTHESIS OF 2-THIOHISTIDINE AND THE LIKE TETRAHEDRON (FR) 2015-03-25 EP disclosed
US-8835477-B2 Method for the synthesis of 2-thiohistidine and the like TETRAHEDRON (FR) 2014-09-16 US disclosed
US-8835477-B2 Method for the synthesis of 2-thiohistidine and the like TETRAHEDRON (FR) 2014-09-16 US disclosed
US-8399500-B2 Method of synthesizing ergothioneine and analogs TETRAHEDRON (FR) 2013-03-19 US disclosed
US-20120330029-A1 METHOD FOR THE SYNTHESIS OF 2-THIOHISTIDINE AND THE LIKE TETRAHEDRON (FR) 2012-12-27 US disclosed
US-20120330029-A1 METHOD FOR THE SYNTHESIS OF 2-THIOHISTIDINE AND THE LIKE TETRAHEDRON (FR) 2012-12-27 US disclosed
US-20120136159-A1 THE METHOD OF SYNTHESIZING ERGOTHIONEINE AND ANALOGS TERTRAHEDRON (FR) 2012-05-31 US disclosed
WO-2011042480-A1 METHOD FOR THE SYNTHESIS OF ERGOTHIONEINE AND THE LIKE TETRAHEDRON (FR) 2011-04-14 WO disclosed
WO-2011042478-A1 METHOD FOR THE SYNTHESIS OF 2-THIOHISTIDINE AND THE LIKE TETRAHEDRON (FR) 2011-04-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120136159-A1 THE METHOD OF SYNTHESIZING ERGOTHIONEINE AND ANALOGS TST, SLC6A12, TTPA SLC22A4 331/4885KDM3B 4522/4885ITGB2 4352/4885
US-20120330029-A1 METHOD FOR THE SYNTHESIS OF 2-THIOHISTIDINE AND THE LIKE TST, CTH, TPMT SLC22A4 1293/4885KDM3B 3157/4885ITGB2 3730/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.