SCHEMBL9622893

SCHEMBL9622893

C[C@]12CCCC=C1CC[C@@H]1C2=CC[C@@]2(C)[C@H]1CC[C@]2(O)C#N

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 3/20 0.41
AR P10275 2/20 0.41
PGR P06401 2/20 0.41
NR3C2 P08235 1/20 0.41
CYP19A1 P11511 14/20 0.38
ABCB11 O95342 1/20 0.37
MAOA P21397 1/20 0.35
OPRK1 P41145 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HIF1A Q16665 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10582213 1.00 NR3C1 (0.41) NR3C1ARPGRNR3C2CYP19A1
SCHEMBL9623805 0.83 NR3C1 (0.60) NR3C1ARPGRNR3C2CYP19A1
SCHEMBL8940232 0.83 NR3C1 (0.60) NR3C1ARPGRNR3C2CYP19A1
SCHEMBL9623872 0.81 NR3C1 (0.45) NR3C1ARPGRNR3C2CYP19A1
SCHEMBL9470387 0.81 ESR1 (0.46) NR3C1ARPGRNR3C2CYP19A1
SCHEMBL8939564 0.75 NR3C1 (0.40) NR3C1ARPGRNR3C2CYP19A1
SCHEMBL9623669 0.75 NFKB1 (0.56) NR3C1ARPGRNR3C2CYP19A1
SCHEMBL10724042 0.74 NR3C1 (0.38) NR3C1ARPGRNR3C2CYP19A1
SCHEMBL11639279 0.73 CYP19A1 (0.43) NR3C1CYP19A1
SCHEMBL10413728 0.72 NR3C1 (0.58) NR3C1ARPGRNR3C2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0153001-B1 STEROIDS HAVING AN ENAMIDE OR ENIMIDE GROUP AND THEIR PREPARATION THE UPJOHN COMPANY (US) 1992-03-11 EP disclosed
US-4831131-A 11β,17α-Dihydroxy-17β-cyano-androstanes THE UPJOHN COMPANY (US) 1989-05-16 US disclosed
US-4585590-A Cyanohydrin process THE UPJOHN COMPANY (US) 1986-04-29 US disclosed
US-4548748-A Cyanohydrin process THE UPJOHN COMPANY (US) 1985-10-22 US disclosed
EP-0153001-A2 Steroids having an enamide or enimide group and their preparation THE UPJOHN COMPANY (US) 1985-08-28 EP disclosed
US-4500461-A Cyanohydrin process THE UPJOHN COMPANY (US) 1985-02-19 US disclosed