SCHEMBL9624802

SCHEMBL9624802

Cc1cccc2c(CCN(C)CCCN3Cc4cc5c(cc4C3=O)OCO5)c[nH]c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.40
HTR2A P28223 2/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
HTR1A P08908 1/20 0.37
HTR1D P28221 1/20 0.37
HTR1B P28222 1/20 0.37
HTR2C P28335 1/20 0.37
HTR1E P28566 1/20 0.37
HTR1F P30939 1/20 0.37
HTR7 P34969 1/20 0.37
HTR2B P41595 1/20 0.37
HTR3A P46098 1/20 0.37
HTR5A P47898 1/20 0.37
HTR6 P50406 1/20 0.37
HTR4 Q13639 1/20 0.37
HTR3D Q70Z44 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624504 0.90 HTR2A (0.43) DRD2HTR2AMAPTSMN1; SMN2NPSR1
SCHEMBL9624748 0.88 BCHE (0.44) DRD2HTR2AMAPTNPSR1HTR3E
SCHEMBL9624887 0.86 HTR6 (0.45) HTR2AMAPTSMN1; SMN2NPSR1HTR6
SCHEMBL9624496 0.85 KMT2A (0.46) DRD2HTR2AMAPTHTR3EHTR3B
SCHEMBL9625146 0.82 SLC6A4 (0.46) DRD2HTR2AHTR3EHTR3BHTR1A
SCHEMBL9625049 0.81 HTR1A (0.49) HTR2AMAPTSMN1; SMN2HTR3EHTR3B
SCHEMBL9625131 0.80 SIGMAR1 (0.35)
SCHEMBL9623773 0.80 BCHE (0.46) DRD2HTR2AMAPTSMN1; SMN2HTR1A
SCHEMBL9625186 0.79 SMPD1 (0.34) MAPT
SCHEMBL9624939 0.78 HTR1D (0.54) MAPTSMN1; SMN2HTR1DHTR6KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
EP-0269968-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-06-08 EP disclosed