SCHEMBL9628948

SCHEMBL9628948

CCCNCC1COc2ccc(OC)cc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.55
HTR2B P41595 2/20 0.44
SIGMAR1 Q99720 2/20 0.44
DRD2 P14416 1/20 0.42
DRD3 P35462 1/20 0.42
POLB P06746 1/20 0.42
ESR2 Q92731 1/20 0.42
MTNR1A P48039 5/20 0.41
HTR7 P34969 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
CYP3A4 P08684 3/20 0.40
MEN1 O00255 2/20 0.40
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
USP2 O75604 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24090506 0.82 HTR2B (0.55) HTR1AHTR2BSIGMAR1DRD2DRD3
Methylamine SCHEMBL10700891 0.80 HTR1A (0.50) HTR1AHTR2BSIGMAR1DRD2DRD3
SCHEMBL9629898 0.79 MTNR1A (0.56) MTNR1A
SCHEMBL9627798 0.77 HTR1A (0.50) HTR1AHTR2BSIGMAR1DRD2DRD3
SCHEMBL9628106 0.77 PPARD (0.56)
SCHEMBL9627910 0.76 HTR1A (0.44) HTR1AHTR2BSIGMAR1DRD2DRD3
SCHEMBL9628688 0.75 HTR2B (0.43) HTR1AHTR2BSIGMAR1DRD2DRD3
SCHEMBL172889 0.75 HTR1A (0.57) HTR1AHTR2BSIGMAR1DRD2DRD3
SCHEMBL135119 0.75 MTNR1A (0.65) MTNR1A
SCHEMBL10692134 0.74 HTR1A (0.43) HTR1AHTR2BSIGMAR1DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0281261-B1 3-AMINOMETHYL DERIVATIVES OF INDANE, INDOLINE AND DIHYDROBENZOFURANE AND DIHYDROBENZOTHIOPHENE H. LUNDBECK A/S (DK) 1992-05-06 EP disclosed
US-4946863-A CNS-affecting 6-oxy-3-aminomethyl indanes, compositions thereof, and method of treating therewith H. LUNDBECK A/S (DK) 1990-08-07 US disclosed
US-4847254-A CNS affecting 5-oxy-3-aminomethyl-dihydro-benzofurans and benzothiophenes H. LUNDBECK A/S (DK) 1989-07-11 US disclosed
EP-0281261-A2 3-Aminomethyl derivatives of indane, indoline and dihydrobenzofurane and dihydrobenzothiophene H. LUNDBECK A/S (DK) 1988-09-07 EP disclosed